| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
US10040781, Example 242 |
NA |
249000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 245 |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 495 |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 487 |
NA |
324000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((3-fluoro-4-(piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(((3R,4S)-3-fluorotetrahydro-2H-pyran-4-yl)oxy)benzonitrile |
NA |
373000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 362 |
NA |
747000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-(2-oxo-2,3-dihydrooxazole-4-carbonyl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 434 |
NA |
865000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 493 |
NA |
782000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
(R)-2-((1-(2-hydroxyacetyl)piperidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
952000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((4-(tetrahydro-2H-pyran-4-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 252 |
NA |
213000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 246 |
NA |
181000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluorotetrahydro-2H-pyran-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
397000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((2-(2-hydroxypropan-2-yl)pyridin-4-yl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 381 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 593 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 604 |
NA |
950000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 600 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 597 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |