| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK3 |
4-amino-N-benzyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| JAK3 |
|
8700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-[2-Benzyloxy-5-(4-isobutoxybenzoyl)phenyl]propionic acid |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-[2-Isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propionic acid |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-[2-Isobutoxy-5-(4-propoxybenzoyl)phenyl]propionic acid |
NA |
930000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
(R)-4-(4-methylpentanoyl)-8-(4-methylpentylidene)-1-thia-4-azaspiro[4.5]decane-3-carboxylic acid |
NA |
650000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
(R)-8-(3-methylbutylidene)-4-(5-methylhexanoyl)-1-thia-4-aza-spiro[4.5]decane-3-carboxylic acid |
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-[5-(4-Isobutoxybenzoyl)-2-propoxyphenyl]propionic acid |
NA |
910000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-[2-Isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propionic acid |
NA |
610000 |
NA |
NA |
NA |
NA |
BindingDB |
| JUN |
3-(4-Chloro-phenyl)-2-(2-methylamino-4-phenyl-thiazol-5-yl)-3H-quinazolin-4-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| JUN |
(1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
NA |
480000 |
NA |
NA |
NA |
NA |
PubChem |
| JUN |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
1000000 |
NA |
PubChem |
| KARS1 |
3-O-(1-benzhydrylazetidin-3-yl) 5-O-propan-2-yl 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
Cladosporin |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
NA |
286000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
Azelastine |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
3-Methyl 5-(1-(phenylmethyl)-3-piperidinyl) 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylate |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
Manidipine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
Nisoldipine |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB |
| KARS1 |
Cilnidipine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |