| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KAT2B |
5-Hydroxymethyl-2-phenylisothiazol-3(2H)-one |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KAT2B |
5-Acetoxymethyl-2-phenylisothiazol-3(2H)-one |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KAT2B |
Ac-Lys(CoA)-NH2 |
NA |
108300|200000 |
NA |
NA |
NA |
NA |
BindingDB|GtoPDB|TTD |
| KAT2B |
(Z)-2-Hydroxy-6-(4-(pentyloxy)styryl)benzoic acid |
NA |
662000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KAT2B |
2-[[4-(Trifluoromethyl)phenyl]methyl]-[1,2]thiazolo[5,4-b]pyridin-3-one |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT2B |
2-[(3,4-Difluorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-one |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KAT2B |
[[(3S)-4-[[3-[2-[[1-[(5S)-5-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamidopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[(2S)-1-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-6-oxohexyl]triazol-4-yl]methylsulfanyl]ethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphate |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT2B |
Ac-SGRGKGGK(CoA)GLGKGGAKRHRK |
NA |
124300 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT2B |
2-Hydroxy-6-(8Z,11Z)-8,11,14-pentadecatrien-1-ylbenzoic acid |
NA |
667050|1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KAT5 |
US11911372, Example 83 |
NA |
108630 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
US11911372, Example 81 |
NA |
121010 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
N-(5-phenylisoxazol-3-yl)propane-1-sulfonamide |
NA |
116160 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
4-methoxy-N-(5-phenylisoxazol-3-yl)benzenesulfonamide |
NA |
113950 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
US11492346, Example 26 |
125000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
2-[4-[2-[3-(3,4-Dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-1,3-thiazol-4-yl]phenyl]isoindole-1,3-dione |
NA |
149000 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
(1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| KAT5 |
Ac-SGRGK(CoA)GGKGLGKGGAKRHRK |
NA |
143350 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
Ac-SGRGKGGK(CoA)GLGKGGAKRHRK |
NA |
111700 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT5 |
2-Hydroxy-6-(8Z,11Z)-8,11,14-pentadecatrien-1-ylbenzoic acid |
NA |
374590 |
NA |
NA |
NA |
NA |
BindingDB |
| KAT6A |
3-chloro-N-(5-phenylisoxazol-3-yl)benzenesulfonamide |
NA |
109990 |
NA |
NA |
NA |
NA |
BindingDB |