| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MGAM |
(S)-3-(2-((4aR,6aS,7R,10aS,10bR)-6a,10b-dimethyl-8-methylene-3-phenyl-decahydro-1H-naphtho[2,1-d][1,3]dioxin-7-yl)ethylidene)-4-hydroxy-dihydrofuran-2(3H)-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| MGAM |
Precose |
NA |
906000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| MGAM |
Validamine |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| MGAM |
N-[5-(Adamantan-1-yl-methoxy)-pentyl]-L-altro-1-deoxynojirimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MGAM |
3,4-Pyrrolidinediol, 2-(hydroxymethyl)-1-methyl-, (2R,3R,4R)- |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGAM2 |
1-Deoxynojirimycin |
NA |
192000 |
NA |
NA |
NA |
NA |
PubChem |
| MGAM2 |
Glucobay |
NA |
189200|420200|817000|583600|707900|442400|101500|817380|320000|942000|576200|1520000|452243|200800 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| MGEA5 |
N-[(2S,3R,4R,5S,6R)-2-[6-[4-[(1,3-dioxobenzo[de]isoquinolin-2-yl)methyl]triazol-1-yl]hexylsulfanyl]-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]acetamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
1-[4-[4-(4-Fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]-2-phenylethanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
4-benzhydryl-N-phenylpiperazine-1-carbothioamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
5-{4-nitrobenzoyl}-2-(3-pyridinyl)-1H-isoindole-1,3(2H)-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
4-chloro-N-(2-phenylethyl)benzenecarbothioamide |
NA |
436516|436515.83 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MGLL |
2-[[5-(4-Methoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-[4-(4-methoxyphenyl)piperazin-1-yl]ethanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
(3-Chlorophenyl)(morpholino)methanethione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
Methyl diethyldithiocarbamate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
(Diethylcarbamoyl)methylene diethylcarbamodithioate |
NA |
630957.34 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MGLL |
3,4-dihydroxy-N-(2-phenylethyl)benzenecarbothioamide |
NA |
524807|524807.46 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MGLL |
2-[5-(4-Morpholin-4-ylphenyl)tetrazol-2-yl]-1-(4-phenylpiperazin-1-yl)ethanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
1-[4-(4-Fluorophenyl)piperazin-1-yl]-2-[5-(4-methoxyphenyl)tetrazol-2-yl]ethanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MGLL |
[1-Phenyl-5-(4-phenylmethoxyphenyl)pyrazol-3-yl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |