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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MGLL (+/-)-3-(But-3-enyl)-1-pent-4-enoylazetidin-2-one NA 817000 NA NA NA NA BindingDB|TTD
MGLL 1-(Benzotriazol-1-yl)-2-[4-(2-methylpropyl)phenyl]propan-1-one NA 194984.46 NA NA NA NA TTD
MGLL Ibuproxam, dimethyl deriv. NA 645654.23 NA NA NA NA TTD
MGLL 3-[4-(2-Methylpropyl)phenyl]-1-nitrobutan-2-one NA 489778.82 NA NA NA NA TTD
MGLL 1-Chloro-3-[4-(2-methylpropyl)phenyl]butan-2-one NA 199526.23 NA NA NA NA TTD
MGLL (2,4-Dichlorophenyl)(morpholino)methanethione NA 1000000 NA NA NA NA TTD
MGLL Methyl morpholine-4-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL 2-Octyl-1,2-benzoxazol-3-one NA 275000 NA NA NA NA BindingDB|TTD
MGLL 2-(4-Benzhydrylpiperazin-1-yl)-1-phenyl-2-sulfanylideneethanone NA 1000000 NA NA NA NA TTD
MGLL Phenyl 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (4-Methylphenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (4-Chlorophenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (2-Chlorophenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (4-Methoxyphenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (4-Acetylphenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL (4-Tert-butylphenyl) 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL [4-(Trifluoromethyl)phenyl] 4-benzhydrylpiperazine-1-carbodithioate NA 1000000 NA NA NA NA TTD
MGLL 2,3-bis(furan-3-yl)-N-[(4-methoxyphenyl)methyl]quinoxaline-6-carboxamide NA 500000 NA NA NA NA TTD
MGLL (4-(Dimethylamino)phenyl)(morpholino)methanethione NA 1000000 NA NA NA NA TTD
MGLL Morpholine, 4-(phenylthioacetyl)- NA 1000000 NA NA NA NA TTD