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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MGMT 6-pentoxy-7H-purin-2-amine NA 1006000 NA NA NA NA BindingDB|TTD
MGMT O6-Substituted Guanine Deriv. 11 NA 1000000 NA NA NA NA TTD
MGMT O6-Substituted Guanine Deriv. 18 NA 1000000 NA NA NA NA TTD
MGMT O6-Substituted Guanine Deriv. 21 NA 192000 NA NA NA NA BindingDB
MGMT 6-(cyclopentylmethoxy)-9H-purin-2-amine NA 1000000 NA NA NA NA TTD
MGMT O6-Substituted Guanine Deriv. 27 NA 1000000 NA NA NA NA TTD
MGMT 6-(2-Phenylethoxy)-9H-purin-2-amine NA 548000 NA NA NA NA BindingDB|TTD
MGMT O6-Substituted Guanine Deriv. 41 NA 1000000 NA NA NA NA TTD
MGMT O6-Substituted Guanine Deriv. 42 NA 1000000 NA NA NA NA TTD
MGMT 2-Amino-4-benzyloxy-6-[N-(4-(4-aminophenoxy)anilino)]-5-nitropyrimidine NA 600000 NA NA NA NA TTD
MGMT 2-Amino-4-benzyloxy-6-[N-(4,4''-diaminobenzophenone)]-5-nitropyrimidine NA 600000 NA NA NA NA TTD
MGMT O-(6)-Methylguanine NA 248000|428000 NA NA NA NA BindingDB|TTD
MGMT Purine, 2-amino-6-propoxy- NA 1000000 NA NA NA NA TTD
MGMT 6-butoxy-9H-purin-2-amine NA 493000 NA NA NA NA BindingDB|TTD
MGMT 6-Ethylguanine NA 1000000 NA NA NA NA TTD
MIF Porphobilinogen NA 400000 NA NA NA NA PubChem
MIF (E)-2-(2-Hydroxybenzylidene)-3,4-dihydronaphthalen-1(2H)-one NA 1158000 NA NA NA NA BindingDB
MIF 2,6-dimethoxy-N-((5-(thiophen-2-yl)-1,3,4-oxadiazol-2-yl)methyl)benzamide NA 199526 NA NA NA NA BindingDB
MIF 4-Hydroxybenzaldehyde methyl(phenyl)hydrazone NA 300000 NA NA NA NA TTD
MIF [(E)-(4-hydroxyphenyl)methylideneamino] 2,2-dimethylpropanoate NA 113000 NA NA NA NA TTD