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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MGLL N-(2-phenylethyl)benzenecarbothioamide NA 1000000 NA NA NA NA TTD
MGLL [(1R)-1-[(3S)-2-oxo-1-(prop-2-enylcarbamothioyl)azetidin-3-yl]ethyl] 2-phenylmethoxyacetate NA 121700 NA NA NA NA BindingDB|TTD
MGLL 2-chloro-N-(2-phenylethyl)benzenecarbothioamide NA 165959|165958.69 NA NA NA NA BindingDB|TTD
MGLL (4-Cyclohexylphenyl)-morpholin-4-ylmethanethione NA 1000000 NA NA NA NA TTD
MGLL N-(2-phenylethyl)-2-(4-phenylphenyl)ethanethioamide NA 537032|537031.8 NA NA NA NA BindingDB|TTD
MGLL 2-(3,4-Dimethoxy-phenyl)-1-morpholin-4-yl-ethanethione NA 1000000 NA NA NA NA TTD
MGLL 4-(Biphenyl-4-ylmethyl)morpholine NA 1000000 NA NA NA NA TTD
MGLL 4-(2-Chlorobenzyl)morpholine NA 1000000 NA NA NA NA TTD
MGLL 4-[(4-Chlorophenyl)methyl]morpholine NA 1000000 NA NA NA NA TTD
MGLL (3,4-Dichlorophenyl)(morpholino)methanethione NA 1000000 NA NA NA NA TTD
MGMT 2,6-Diamino-4-(benzyloxy)pyrimidine NA 170000 NA NA NA NA BindingDB|TTD
MGMT 6-Hex-3-enyloxy-9H-purin-2-ylamine NA 1000000 NA NA NA NA TTD
MGMT 1-(2-Amino-9H-purin-6-yloxy)-butan-2-one NA 151000 NA NA NA NA BindingDB
MGMT 6-(2,2-Dimethyl-[1,3]dioxolan-4-ylmethoxy)-9H-purin-2-ylamine NA 1000000 NA NA NA NA TTD
MGMT 6-(2,2-Dimethoxy-2-phenyl-ethoxy)-9H-purin-2-ylamine NA 1000000 NA NA NA NA TTD
MGMT 2-(2-Amino-9H-purin-6-yloxy)-1-phenyl-ethanone NA 1000000 NA NA NA NA TTD
MGMT 6-Hexyloxy-9H-purin-2-ylamine NA 554000 NA NA NA NA BindingDB|TTD
MGMT 6-Cyclobutylmethoxy-9H-purin-2-ylamine NA 1000000 NA NA NA NA TTD
MGMT 1-[(2-Amino-6,9-Dihydro-1h-Purin-6-Yl)Oxy]-3-Methyl-2-Butanol NA 1000000 NA NA NA NA TTD
MGMT 6-O-Cyclohexylmethyl Guanine NA 1000000 NA NA NA NA TTD