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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MGLL 1-phenyl-5-(4-phenylmethoxyphenyl)-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]pyrazole-3-carboxamide NA 200000 NA NA NA NA TTD
MGLL [5-(4-Hydroxyphenyl)-1-methylpyrazol-3-yl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone NA 132000 NA NA NA NA BindingDB|TTD
MGLL N-(1-benzylpiperidin-4-yl)-5-(4-hydroxyphenyl)-1-phenylpyrazole-3-carboxamide NA 200000 NA NA NA NA TTD
MGLL 5-(4-hydroxyphenyl)-1-phenyl-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]pyrazole-3-carboxamide NA 200000 NA NA NA NA TTD
MGLL 4-(3-fluoro-4-methoxyphenyl)-2-[(E)-N-hydroxy-C-pentadecylcarbonimidoyl]phenol NA 200000 NA NA NA NA TTD
MGLL 2-[(E)-C-butyl-N-hydroxycarbonimidoyl]-4-(4-methoxyphenyl)phenol NA 119000 NA NA NA NA BindingDB|TTD
MGLL 4-(3-fluoro-4-methoxyphenyl)-2-[(E)-N-hydroxy-C-tridecylcarbonimidoyl]phenol NA 200000 NA NA NA NA TTD
MGLL Morpholine-4-carbothioylsulfanylmethyl morpholine-4-carbodithioate NA 102329.3 NA NA NA NA BindingDB|TTD
MGLL Thiobenzoylmorpholine NA 1000000 NA NA NA NA TTD
MGLL 4-fluoro-N-(2-phenylethyl)benzenecarbothioamide NA 1000000 NA NA NA NA TTD
MGLL (3-Methylphenyl)-piperidin-1-ylmethanethione NA 1000000 NA NA NA NA TTD
MGLL ST043087 NA 1000000 NA NA NA NA TTD
MGLL 4-(2-Chlorobenzoyl)-morpholine NA 1000000 NA NA NA NA TTD
MGLL N-(4-Chlorobenzoyl)morpholine NA 1000000 NA NA NA NA TTD
MGLL 1-Pent-4-enoyl-3-(pent-4-enyl)azetidin-2-one NA 657000 NA NA NA NA BindingDB|TTD
MGLL 1-(Phenylthioxomethyl)piperidine NA 1000000 NA NA NA NA TTD
MGLL 4-(4-Hydroxythiobenzoyl)morpholine NA 204174|204173.79 NA NA NA NA BindingDB|TTD
MGLL N-(4-acetylphenyl)-1-(4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxamide NA 500000 NA NA NA NA TTD
MGLL [(1R)-1-[(2R,3R)-2-acetyloxy-4-oxo-1-pent-4-enoylazetidin-3-yl]ethyl] pent-4-enoate NA 133000 NA NA NA NA BindingDB|TTD
MGLL (2-Morpholin-4-yl-2-oxoethyl) morpholine-4-carbodithioate NA 218776.16 NA NA NA NA BindingDB|TTD