| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MT-CO1 |
2-[3-(4-Fluorophenyl)-6-oxo-4,5-dihydropyridazin-1-yl]-4-(4-methoxyphenyl)-1-methyl-6-oxopyrimidine-5-carbonitrile |
NA |
115260 |
NA |
NA |
NA |
NA |
BindingDB |
| MT-CO2 |
1-(4-Bromophenyl)-3-(2-oxocyclohexyl)pyrrolidine-2,5-dione |
NA |
113440 |
NA |
NA |
NA |
NA |
BindingDB |
| MTNR1A |
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[2-(2-hydroxy-5-prop-2-enylphenyl)-4-prop-2-enylphenoxy]oxane-3,4,5-triol |
NA |
NA |
NA |
396500 |
NA |
NA |
BindingDB|TTD |
| MTNR1A |
Bisphenol F |
NA |
NA |
NA |
237000 |
NA |
NA |
BindingDB|TTD |
| MTNR1A |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]pyrrolidine |
NA |
NA |
NA |
310000 |
NA |
NA |
BindingDB |
| MTNR1A |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]piperazine |
NA |
NA |
NA |
460000 |
NA |
NA |
BindingDB |
| MTNR1A |
(5-Methoxy-6-methyl-1-benzofuran-3-yl)methanol |
NA |
NA |
NA |
700000 |
NA |
NA |
BindingDB |
| MTNR1A |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]-4-methylpiperazine |
NA |
NA |
NA |
330000 |
NA |
NA |
BindingDB |
| MTNR1A |
1-(5-methoxy-6-methyl-1-benzofuran-3-yl)-N,N-dimethylmethanamine |
NA |
NA |
NA |
440000 |
NA |
NA |
BindingDB |
| MTNR1A |
(5-Methoxy-6-methyl-1-benzofuran-3-yl)methanamine |
NA |
NA |
NA |
250000 |
NA |
NA |
BindingDB |
| MTNR1A |
1,4-Bis[(5-methoxy-6-methyl-1-benzofuran-3-yl)methyl]piperazine |
NA |
NA |
NA |
420000 |
NA |
NA |
BindingDB |
| MTNR1A |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]-4-methyl-1,4-diazepane |
NA |
NA |
NA |
380000 |
NA |
NA |
BindingDB |
| MTNR1A |
N-ethyl-N-[(5-methoxy-6-methyl-1-benzofuran-3-yl)methyl]ethanamine |
NA |
NA |
NA |
360000 |
NA |
NA |
BindingDB |
| MTNR1A |
epicatechin-(4beta->8)-4'-O-methylgallocatechin |
NA |
156100 |
NA |
NA |
NA |
NA |
BindingDB |
| MTNR1A |
Agomelatine |
NA |
NA |
NA |
5800000 |
NA |
NA |
BindingDB|PubChem |
| MTNR1B |
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[2-(2-hydroxy-5-prop-2-enylphenyl)-4-prop-2-enylphenoxy]oxane-3,4,5-triol |
NA |
NA |
NA |
383000 |
NA |
NA |
BindingDB|TTD |
| MTNR1B |
N-[3-(5-methoxy-1H-indol-2-yl)propyl]acetamide |
102329|102329.3 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MTNR1B |
Bisphenol F |
NA |
NA |
NA |
244000 |
NA |
NA |
BindingDB|TTD |
| MTNR1B |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]pyrrolidine |
NA |
NA |
NA |
350000 |
NA |
NA |
BindingDB |
| MTNR1B |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]piperazine |
NA |
NA |
NA |
380000 |
NA |
NA |
BindingDB |