| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MTOR |
5-[2-[(4-Methylsulfonylpiperazin-1-yl)methyl]-8-morpholin-4-ylimidazo[1,2-a]pyrazin-6-yl]-4-(trifluoromethyl)pyrimidin-2-amine |
NA |
10000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MTOR |
Benzenesulfonanilide |
NA |
NA |
1000000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
6-Hydroxy-4-methyl-2-benzopyrone |
NA |
NA |
760000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
4-Carbethoxy-3-methyl-2-cyclohexen-1-one |
NA |
NA |
410000 |
NA |
NA |
NA |
BindingDB |
| MVD |
(2R)-1-[2-[hydroxy(phosphonooxy)phosphoryl]oxyacetyl]pyrrolidine-2-carboxylic acid |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| MYC |
N-2-Biphenylyl-7-nitro-2,1,3-benzoxadiazol-4-amine |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYC |
Mefenamic Acid |
NA |
403000 |
NA |
NA |
NA |
NA |
PubChem |
| MYLK |
1-[4-(4-chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
10900000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 4-(4-chlorophenyl)-2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
5490000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(2-chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
10200000|10204224.39 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYLK |
1-[4-(4-fluorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
13600000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(2-hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
23200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
23700000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
46700000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[2-methyl-4-(3-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
49000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[2-methyl-4-(4-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
49000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-[4-(dimethylamino)phenyl]-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
22800000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-hydroxy-3-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]ethanone |
NA |
27200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(2-chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
9250000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-chlorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
9000000 |
NA |
NA |
NA |
NA |
BindingDB |