| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MYLK |
1-[4-(4-fluorophenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
7510000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(2-hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
21200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-hydroxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
16900000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
46000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[2-methyl-4-(3-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
47600000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[2-methyl-4-(4-nitrophenyl)-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
32800000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-[4-(dimethylamino)phenyl]-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
13500000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
1-[4-(4-hydroxy-3-methoxyphenyl)-2-methyl-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl]propan-1-one |
NA |
27200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
N-(2-guanidinoethyl)-5-isoquinolinesulfonamide |
150000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYLK |
ethyl 2-methoxy-6-methyl-3-phenacyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
4290000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-4-phenyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
7510000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 4-(4-chlorophenyl)-2-methoxy-6-methyl-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
3190000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 4-(4-chlorophenyl)-3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
2420000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-4-(4-methoxyphenyl)-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
3300000|3300350.01 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYLK |
ethyl 4-(4-hydroxyphenyl)-2-methoxy-6-methyl-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
9800000|9803925.45 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYLK |
ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-4-(4-hydroxyphenyl)-2-methoxy-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
6570000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 4-(4-hydroxyphenyl)-2-methoxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-6-methyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
10200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MYLK |
ethyl 2-methoxy-6-methyl-4-(4-methylphenyl)-3-phenacyl-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
5200000|5208348.07 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MYLK |
ethyl 3-[2-(4-chlorophenyl)-2-oxoethyl]-2-methoxy-6-methyl-4-(4-methylphenyl)-2,4-dihydro-1H-pyrimidine-5-carboxylate |
NA |
3420000 |
NA |
NA |
NA |
NA |
BindingDB |