| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(aminomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[2-(3,4-dichlorophenyl)ethyl]acetamide |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[2-[3-(trifluoromethyl)phenyl]ethyl]acetamide |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[2-(4-chlorophenyl)ethyl]acetamide |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[2-(1-methylindol-3-yl)ethyl]acetamide |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-prop-2-ynylacetamide |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-[(dimethylsulfamoylamino)methyl]-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[2-(3,4-dichlorophenyl)ethyl]acetamide |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-[(2-chloropyridin-4-yl)methyl]acetamide |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
2-[6-amino-9-[(2R,3R,4S,5R)-5-(azidomethyl)-3,4-dihydroxyoxolan-2-yl]purin-8-yl]sulfanyl-N-(3-phenylpropyl)acetamide |
150000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
(Tiazofurin-5''-yl)(adenosin-5''-yl)disulfide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| NADK |
Di(2''-C-methyladenosine-5''-yl)disulfide |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
| NAE1 |
Candesartan Cilexetil |
NA |
NA |
195000 |
NA |
NA |
NA |
PubChem |
| NALCN |
Verapamil |
NA |
380000 |
NA |
NA |
NA |
NA |
GtoPDB |
| NAMPT |
2-[(2-fluorophenyl)amino]-6-propylpyrimidin-4(3H)-one |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| NAMPT |
3-(2-Pyridin-2-ylethyl)-3-azabicyclo[3.2.0]heptane-2,4-dione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NAMPT |
5-methyl-1-phenyl-N-(pyridin-3-yl)-1H-pyrazole-4-carboxamide |
NA |
NA |
177000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| NAMPT |
Diazoxide |
NA |
NA |
230000 |
NA |
NA |
NA |
BindingDB|ChEMBL|PubChem |
| NAMPT |
1-Ethyl-3-methyl-N-(pyridin-3-yl)-1H-pyrazole-4-carboxamide |
NA |
NA |
233000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| NAMPT |
3-methyl-N-(pyridin-3-yl)thiophene-2-carboxamide |
NA |
NA |
129000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| NAMPT |
1-(3,4-Difluorophenyl)-3-(pyridin-4-ylmethyl)urea |
NA |
850000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| NAMPT |
N-pyridin-3-yl-1H-pyrazole-5-carboxamide |
NA |
NA |
176000 |
NA |
NA |
NA |
BindingDB|ChEMBL |