| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MTNR1B |
(5-Methoxy-6-methyl-1-benzofuran-3-yl)methanol |
NA |
NA |
NA |
520000 |
NA |
NA |
BindingDB |
| MTNR1B |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]-4-methylpiperazine |
NA |
NA |
NA |
260000|298900 |
NA |
NA |
BindingDB |
| MTNR1B |
1-(5-methoxy-6-methyl-1-benzofuran-3-yl)-N,N-dimethylmethanamine |
NA |
NA |
NA |
130000 |
NA |
NA |
BindingDB |
| MTNR1B |
(5-Methoxy-6-methyl-1-benzofuran-3-yl)methanamine |
NA |
NA |
NA |
350000 |
NA |
NA |
BindingDB |
| MTNR1B |
1,4-Bis[(5-methoxy-6-methyl-1-benzofuran-3-yl)methyl]piperazine |
NA |
NA |
NA |
430000 |
NA |
NA |
BindingDB |
| MTNR1B |
1-[(5-Methoxy-6-methyl-1-benzofuran-3-yl)methyl]-4-methyl-1,4-diazepane |
NA |
NA |
NA |
270000 |
NA |
NA |
BindingDB |
| MTNR1B |
N-ethyl-N-[(5-methoxy-6-methyl-1-benzofuran-3-yl)methyl]ethanamine |
NA |
NA |
NA |
360000 |
NA |
NA |
BindingDB |
| MTNR1B |
epicatechin-(4beta->8)-4'-O-methylgallocatechin |
NA |
208800 |
NA |
NA |
NA |
NA |
BindingDB |
| MTNR1B |
Agomelatine |
NA |
NA |
NA |
17300000 |
NA |
NA |
BindingDB|PubChem |
| MTOR |
4-[4-[6-Bromo-4-(trifluoromethyl)pyridin-3-yl]-6-morpholin-4-yl-1,3,5-triazin-2-yl]morpholine |
660000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MTOR |
4-[4-[6-Chloro-4-(trifluoromethyl)pyridin-3-yl]-6-morpholin-4-yl-1,3,5-triazin-2-yl]morpholine |
NA|110000 |
1100000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MTOR |
1H-1,2,4-Triazole, 5-phenyl- |
NA |
NA |
4000000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
N-Cyclohexylbenzenesulfonamide |
NA |
NA |
500000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
2-(pyridin-3-yl)-1H-1,3-benzodiazole |
NA |
NA |
410000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
Caffeine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| MTOR |
3-(4-Morpholino-1-methyl-1H-pyrazolo[3,4-d]pyrimidine-6-yl)phenol |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB |
| MTOR |
2,6-Dioxo-piperidine-4-carbothioic acid S-butyl ester |
NA |
NA |
190000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
6,7-Dihydroxy-4-methylcoumarin |
NA |
NA |
1500000 |
NA |
NA |
NA |
BindingDB |
| MTOR |
5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)-1H-pyridin-2-one |
NA |
17000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MTOR |
7-Diethylamino-4-methylcoumarin |
NA |
NA |
130000 |
NA |
NA |
NA |
BindingDB |