| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NOTUM |
2-(3-chlorophenoxy)-N-pyridin-3-ylacetamide |
NA |
310000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOTUM |
2-Phenoxy-N-(3-pyridinyl)acetamide |
NA |
150000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOTUM |
4-[4-(Hydroxymethyl)triazol-1-yl]benzonitrile |
NA |
270000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOTUM |
[1-(3-Ethoxyphenyl)triazol-4-yl]methanol |
NA |
230000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOTUM |
(1-phenyl-1H-1,2,3-triazol-4-yl)methanol |
NA |
110000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOTUM |
2-(2-methoxyphenoxy)-N-(pyridin-3-yl)acetamide |
NA |
170000 |
NA |
NA |
NA |
NA |
ChEMBL |
| NOX1 |
6-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-2-N-(3,4-dimethylphenyl)-1,3,5-triazine-2,4-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| NOX1 |
2-N-(3,4-dimethylphenyl)-6-[[4-(3-methylphenyl)piperazin-1-yl]methyl]-1,3,5-triazine-2,4-diamine |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| NPBWR1 |
5-(Methylsulfonyl)-2-phenyl-1H-benzo[d]imidazole |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| NPC1 |
Calcimycin |
NA |
NA |
NA |
NA |
290929 |
NA |
PubChem |
| NPC1 |
Catechol |
NA |
NA |
NA |
NA |
115821 |
NA |
PubChem |
| NPC1 |
Dequalinium |
NA |
NA |
NA |
NA |
183564 |
NA |
PubChem |
| NPC1 |
Mitoxantrone |
NA |
NA |
NA |
NA |
115821 |
NA |
PubChem |
| NPC1 |
Idarubicin |
NA |
NA |
NA |
NA |
115821 |
NA |
PubChem |
| NPC1 |
Ouabain |
NA |
NA |
NA |
NA |
115821 |
NA |
PubChem |
| NPC1 |
Nicardipine |
NA |
NA |
NA |
NA |
115821 |
NA |
PubChem |
| NPC1 |
Rotenone |
NA |
NA |
NA |
NA |
290929 |
NA |
PubChem |
| NPR3 |
NPR-C activator 1 |
NA |
NA |
146000 |
NA |
NA |
NA |
BindingDB |
| NPR3 |
tert-butyl (2S)-2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]-2-cyclohexylacetate |
NA |
NA |
NA |
326700 |
NA |
NA |
BindingDB |
| NPR3 |
(2S)-2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]-4-methylpentanoic acid |
NA |
NA |
220000 |
NA |
NA |
NA |
BindingDB |