| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NQO2 |
5,6,7,8-Tetramethoxy-1,4-dimethylquinolin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| NQO2 |
4-Methylquinolin-2-ol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
Cyanidin |
NA |
NA |
NA |
125200 |
NA |
NA |
TTD |
| NR1H2 |
1-(2-Methylnaphthalen-1-yl)ethan-1-one |
153000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
2-Chloro-1,4-dimethoxybenzene |
476000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
6-Bromo-1,4-dihydro-2H-3,1-benzoxazin-2-one |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
4-Chlorophenol |
NA|169000 |
NA |
NA |
514000|NA |
NA |
NA |
PubChem|TTD |
| NR1H2 |
Methyl indole-6-carboxylate |
302000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
tert-Butyl 4,6-dihydropyrrolo(3,4-c)pyrazole-5(1H)-carboxylate |
225000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H2 |
3-Chlorophenol |
NA|184000 |
NA |
NA |
519000|NA |
NA |
NA |
PubChem|TTD |
| NR1H2 |
3-Bromo-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine |
209000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-4-(3-{[2-fluoro-3-(trifluoromethyl)benzyl]oxy}-phenyl)-8-(trifluoromethyl)cinnoline |
NA |
1336000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-4-(3-{[5-chloro-2-(trifluoromethyl)benzyl]oxy}-phenyl)-8-(trifluoromethyl)cinnoline |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
N-[3-(3-Benzyl-8-chlorocinnolin-4-yl)phenyl]-N-[(1-methyl-1H-indol-7-yl)methyl]amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-8-chloro-4-(3-{[5-fluoro-2-(trifluoromethyl)benzyl]oxy}phenyl)cinnoline |
NA |
1191000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-8-chloro-4-(3-{[5-chloro-2-(trifluoromethyl)-benzyl]oxy}phenyl)cinnoline |
NA |
1826000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-4-[3-(benzyloxy)phenyl]-8-chlorocinnoline |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
[3-(3-Benzyl-8-chlorocinnolin-4-yl)phenyl][5-fluoro-2-(trifluoromethyl)benzyl]amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
[3-(8-Chloro-3-phenylcinnolin-4-yl)phenyl][2-chloro-3-(trifluoromethyl)benzyl]amine |
NA |
179000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
3-Benzyl-8-chloro-4-(3-{[2-chloro-5-(trifluoromethyl)-benzyl]oxy}phenyl)cinnoline |
NA |
147000 |
NA |
NA |
NA |
NA |
TTD |