| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NR1H4 |
2-[(1S,2S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylbutyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
102200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S,4R,5R)-5-[[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy]-3-oxo-2-azabicyclo[2.2.1]heptan-2-yl]-4-(7-oxaspiro[3.5]nonan-2-yl)-1,3-benzothiazole-6-carboxylic acid |
NA |
NA |
NA |
100000000 |
NA |
NA |
BindingDB |
| NR1H4 |
4-[[[2-Chloro-4-[[3-(2,6-dichlorophenyl)-5-(1-methylethyl)-4-isoxazolyl]methoxy]phenyl]methyl]amino]-benzeneacetic acid |
NA |
NA |
NA |
940000 |
NA |
NA |
BindingDB |
| NR1H4 |
3-[(1S)-1-(1,6-dimethylbenzimidazol-2-yl)-2-(1-propan-2-ylsulfonylpiperidin-4-yl)ethyl]-1-(4-phenoxyphenyl)imidazolidine-2,4-dione |
NA |
125500 |
NA |
NA |
NA |
NA |
BindingDB |
| NR1H4 |
Coumarin |
NA |
NA |
NA |
NA |
630957 |
NA |
PubChem |
| NR1H4 |
(E)-3-{3-[Cyclohexanecarbonyl-(4''-dimethylamino-biphenyl-4-ylmethyl)-amino]-phenyl}-acrylic acid |
NA |
NA |
NA |
255000 |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
(E)-3-{3-[Cyclohexanecarbonyl-(4-styryl-benzyl)-amino]-phenyl}-acrylic acid |
NA |
NA |
NA |
255000 |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
(E)-3-{3-[(4-Benzo[1,3]dioxol-5-yl-benzyl)-cyclohexanecarbonyl-amino]-phenyl}-acrylic acid |
NA |
NA |
NA |
222000 |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
(1S,2R,5R,7R,9S,10S,11S,16R)-9-hydroxy-1,2,11,15,15-pentamethyl-5-[(2R,4S,5R)-4,5,6-trihydroxy-6-methylheptan-2-yl]-6-oxapentacyclo[8.8.0.02,7.05,7.011,16]octadecan-14-one |
NA |
NA |
NA |
189050 |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
Fexaramine |
NA |
NA |
1220000 |
NA |
NA |
NA |
BindingDB |
| NR1H4 |
trans-4-((2S)-2-cyclohexyl-2-(2-(2,4-dimethoxypyridin-3-yl)-5,6-difluoro-1H-benzo[d]imidazol-1-yl)acetamido)cyclohexanecarboxylic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| NR1H4 |
2-Phenylphenol |
NA |
NA |
NA |
NA |
501187|891251 |
NA |
PubChem |
| NR1I2 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR1I2 |
Limonene, (+/-)- |
NA |
NA |
NA |
NA |
562341 |
NA |
PubChem |
| NR1I2 |
4-(((6-((3-(2,6-Dichlorophenyl)-5-isopropylisoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid |
NA |
NA |
NA |
1282000 |
NA |
NA |
TTD |
| NR1I2 |
Coumarin |
NA |
NA |
NA |
NA |
1258930 |
NA |
PubChem |
| NR1I2 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR1I2 |
Sodium Azide |
NA |
NA |
NA |
NA |
121972 |
NA |
PubChem |
| NR1I2 |
M-Cresol |
NA |
NA |
NA |
NA |
1584890 |
NA |
PubChem |
| NR1I2 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |