| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NR1I2 |
4-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid |
NA |
NA |
NA |
3871000 |
NA |
NA |
TTD |
| NR1I2 |
3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid |
NA |
NA |
NA |
390000 |
NA |
NA |
TTD |
| NR1I2 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR1I2 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR1I2 |
5-cyclopropyl-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine |
NA |
NA |
NA |
250000 |
NA |
NA |
TTD |
| NR1I2 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| NR1I2 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| NR1I2 |
2-Phenylphenol |
NA |
NA |
NA |
NA |
1412540 |
NA |
PubChem |
| NR1I2 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR1I2 |
2,4-Dimethylphenol |
NA |
NA |
NA |
NA |
891251 |
NA |
PubChem |
| NR1I2 |
Diethylene glycol monomethyl ether |
NA |
NA |
NA |
NA |
1584890 |
NA |
PubChem |
| NR2F2 |
[(4S,5R,12S)-1,5,9-trimethyl-11,14,15,16-tetraoxatetracyclo[10.3.1.04,13.08,13]hexadecan-10-yl] 4-(butan-2-ylamino)-4-oxobutanoate |
NA |
468267 |
NA |
NA |
NA |
NA |
BindingDB |
| NR3C1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
Sundaicumone A |
NA |
NA |
NA |
173000 |
NA |
NA |
TTD |
| NR3C1 |
Norursodeoxycholic acid |
NA |
NA |
NA |
105300 |
NA |
NA |
PubChem|TTD |
| NR3C1 |
Valproic Acid |
NA |
NA |
NA |
NA |
891251 |
NA |
PubChem |
| NR3C1 |
Ursodiol |
NA |
NA |
NA |
298700 |
NA |
NA |
PubChem|TTD |
| NR3C1 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
24-Benzyl-3alpha,7beta-hydroxy-5beta-cholanamide |
NA |
NA |
NA |
109500 |
NA |
NA |
TTD |