| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NR1H3 |
3-Benzyl-4-{3-[(1-methyl-1H-indol-2-yl)methoxy]-phenyl}-8-(trifluoromethyl)cinnoline |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
Quinoline, 4-[3-[(1-methyl-1H-indol-7-yl)methoxy]phenyl]-3-(phenylmethyl)-8-(trifluoromethyl)- |
NA |
668000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
1H-Indole-7-methanamine, N-[3-[3-(phenylmethyl)-8-(trifluoromethyl)-4-quinolinyl]phenyl]- |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H3 |
8-Chloro-4-(3-{[5-chloro-2-(trifluoromethyl)benzyl]oxy}phenyl)-3-phenylcinnoline |
NA |
332000 |
NA |
NA |
NA |
NA |
TTD |
| NR1H4 |
(E)-3-(3-{Cyclohexanecarbonyl-[4-((E)-3-ethoxy-propenyl)-benzyl]-amino}-phenyl)-acrylic acid methyl ester |
NA |
NA |
NA |
198000 |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
(2e)-N-Cyclohexyl-N-(Cyclohexylcarbamoyl)-3-(4-Fluorophenyl)prop-2-Enamide |
NA |
263000 |
NA |
NA |
NA |
NA |
BindingDB |
| NR1H4 |
3-[(1S)-2-cyclohexyl-1-(1,6-dimethylbenzimidazol-2-yl)ethyl]-1-(4-phenoxyphenyl)imidazolidine-2,4-dione |
NA |
126100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
(4S,6S)-3,6-dimethyl-1-(2-methylphenyl)-4-(4-phenoxyphenyl)-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| NR1H4 |
(4R,6R)-3,6-dimethyl-1-(2-methylphenyl)-4-(4-phenoxyphenyl)-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| NR1H4 |
(4S,6R)-3,6-dimethyl-1-(2-methylphenyl)-4-(4-phenoxyphenyl)-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| NR1H4 |
(4R,6S)-6-methyl-1-(2-methylphenyl)-4-(4-phenoxyphenyl)-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| NR1H4 |
(4R,6S)-3-methyl-1-(2-methylphenyl)-4-(4-phenoxyphenyl)-6-propyl-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| NR1H4 |
2-[(1S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-3-methylbutyl]-1-methylbenzimidazole-5-carboxylic acid |
NA |
112900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1R)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylpropyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
118500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]propyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
209500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[3-(4-cyclohexyloxyphenyl)-2,5-dioxoimidazolidin-1-yl]-3-methylbutyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
125500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[2,5-dioxo-4-(4-phenoxyphenyl)piperazin-1-yl]-3-methylbutyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
417500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[4,4-dimethyl-2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-3-methylbutyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
104600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylpropyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
174500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NR1H4 |
2-[(1S)-1-[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]-3-methylbutyl]-3-methylbenzimidazole-5-carboxylic acid |
NA |
398800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |