| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NPR3 |
Tert-butyl 2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]acetate |
NA |
NA |
832000 |
NA |
NA |
NA |
BindingDB |
| NPR3 |
(2S)-2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]-3-phenylpropanoic acid |
NA |
NA |
381000 |
NA |
NA |
NA |
BindingDB |
| NPR3 |
(2S)-2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]-N-methoxy-N,4-dimethylpentanamide |
NA |
NA |
1440000 |
NA |
NA |
NA |
BindingDB |
| NPR3 |
N-[4-[[4-[[(2S)-1-hydroxy-4-methylpentan-2-yl]amino]-1,3,5-triazin-2-yl]amino]phenyl]acetamide |
NA |
NA |
1631000 |
NA |
NA |
NA |
BindingDB |
| NPR3 |
tert-butyl (2S)-2-[[4-(4-acetamidoanilino)-1,3,5-triazin-2-yl]amino]-3,3-dimethylbutanoate |
NA |
NA |
201000 |
NA |
NA |
NA |
BindingDB |
| NPY1R |
2-(6-((4,5-Dimethyloxazol-2-yloxy)methyl)-4-morpholinopyridin-2-ylamino)acetonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NPY1R |
N-(6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-4-morpholinopyridin-2-yl)acetamide |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NPY2R |
2-Diphenylacetylamino-5-guanidino-pentanoic acid ((S)-2-hydroxy-1-phenyl-ethyl)-amide |
NA |
540000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NPY2R |
2-Diphenylacetylamino-5-guanidino-pentanoic acid ((R)-carbamoyl-phenyl-methyl)-amide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| NPY2R |
2-Diphenylacetylamino-5-guanidino-pentanoic acid ((R)-1-phenyl-ethyl)-amide |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NPY2R |
N-[4-Guanidino-1-(7-hydroxy-1,3,4,5-tetrahydro-benzo[c]azepine-2-carbonyl)-butyl]-2,2-diphenyl-acetamide |
NA |
247000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NPY2R |
2-Diphenylacetylamino-5-guanidino-pentanoic acid [1-(4-hydroxy-phenyl)-ethyl]-amide |
NA |
575000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NPY5R |
2-Diphenylacetylamino-5-guanidino-pentanoic acid ((R)-carbamoyl-phenyl-methyl)-amide |
NA |
163000 |
NA |
NA |
NA |
NA |
TTD |
| NQO1 |
4-[(E)-[(6-methoxy-2-methylquinolin-4-yl)hydrazinylidene]methyl]phenol |
NA |
133900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NQO1 |
4-chloro-1-methyl-1H-pyrazolo(3,4-d)pyrimidine |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NQO1 |
4,5-dihydro-1H-imidazol-2-yl(10H-indeno[2,3-b]quinoxalin-11-yl)diazene |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| NQO1 |
[(Z)-[2-(diethoxyphosphorylamino)fluoren-9-ylidene]amino]thiourea |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NQO1 |
|
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| NQO2 |
Quinone, 12 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| NQO2 |
5,6,7,8-tetramethoxy-4-methyl-1H-quinolin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |