| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NR3C1 |
24-Phenethyl-3alpha,7beta-dihydroxy-5beta-cholanamide |
NA |
NA |
NA |
109000 |
NA |
NA |
TTD |
| NR3C1 |
24-alpha-Methylbenzyl-3alpha,7beta-dihydroxy-5beta-cholanamide |
NA |
NA |
NA |
123500 |
NA |
NA |
TTD |
| NR3C1 |
(R)-4-((3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydroxy-10,13-dimethylhexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanenitrile |
NA |
NA |
NA |
101000 |
NA |
NA |
TTD |
| NR3C1 |
(S)-2-((3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydroxy-10,13-dimethylhexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)propanenitrile |
NA |
NA |
NA |
130000 |
NA |
NA |
TTD |
| NR3C1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| NR3C1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| NR3C1 |
2-Phenylphenol |
NA |
NA |
NA |
NA |
446684|501187 |
NA |
PubChem |
| NR3C1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| NR3C1 |
2,4-Dimethylphenol |
NA |
NA |
NA |
NA |
398107 |
NA |
PubChem |
| NR3C2 |
Lecanindole B |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| NR3C2 |
Lecanindole D |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| NR3C2 |
(3S)-3-[1-(4-fluorophenyl)indazol-5-yl]-2,2-dimethyl-3-phenyl-N-(1,3,4-thiadiazol-2-yl)propanamide |
NA |
NA |
NA |
5000000 |
NA |
NA |
TTD |
| NR3C2 |
(3R)-3-[1-(4-fluorophenyl)indazol-5-yl]-2,2-dimethyl-3-phenyl-N-(1,3,4-thiadiazol-2-yl)propanamide |
NA |
NA |
NA |
5000000 |
NA |
NA |
TTD |
| NR4A2 |
7-chloro-N-{3-[(diethylamino)methyl]phenyl}quinolin-4-amine |
NA |
NA |
NA |
116000 |
NA |
NA |
BindingDB|ChEMBL |
| NR4A2 |
4-[(7-Chloroquinolin-4-yl)amino]butanoic acid |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| NR4A2 |
6-Chloroquinolin-4-amine |
NA |
NA |
NA |
117000 |
NA |
NA |
BindingDB|ChEMBL |
| NR4A2 |
5-ethyl-1-phenyl-1H-pyrazole-4-carboxylic acid |
NA |
NA |
NA |
134000 |
NA |
NA |
BindingDB |
| NR4A2 |
7-Chloro-4-aminoquinoline |
NA |
NA |
NA |
259000 |
NA |
NA |
BindingDB|ChEMBL |