| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NT5E |
6-(Furan-3-yl)-3-phenyl-[1,2,4]triazolo[4,3-a]pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
6-(Furan-3-yl)-3-(3-methoxyphenyl)-[1,2,4]triazolo[4,3-a]pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[5-(furan-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[4-Ethyl-6-(2-methylpyrazol-3-yl)benzotriazol-1-yl]phenol |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
6-(furan-3-yl)-3-(1H-indol-6-yl)-[1,2,4]triazolo[4,3-a]pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
6-[6-(Furan-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]-1,3-dihydroindol-2-one |
NA |
148000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(Furan-3-yl)benzimidazol-1-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
6-(furan-3-yl)-3-(5-methyl-1H-indazol-6-yl)-[1,2,4]triazolo[4,3-a]pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(Furan-3-yl)indazol-1-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-(6-Pyrazol-1-yl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)phenol |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
1-(1H-indazol-6-yl)-6-[2-(2-methylphenyl)pyrazol-3-yl]benzotriazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
1-(1H-indazol-6-yl)-6-[2-(4-methylphenyl)pyrazol-3-yl]benzotriazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[4-(Benzylamino)-6-(2-methylpyrazol-3-yl)benzotriazol-1-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(Furan-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]benzoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
2-[6-[(3-Phenylbenzoyl)amino]purin-9-yl]acetic acid |
842700 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
N-[3-[6-(furan-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenyl]methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(2H-triazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
178500 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[5-(Furan-3-yl)triazolo[4,5-d]pyrimidin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(1-Methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(1,3-Oxazol-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |