| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NTRK1 |
Amitriptyline |
NA |
NA |
1800000|2100000|2200000 |
NA |
NA |
NA |
BindingDB|PubChem |
| NTRK1 |
2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-Carbonitrile |
NA |
464000 |
NA |
NA |
NA |
NA |
TTD |
| NTRK2 |
2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-Carbonitrile |
NA |
1190000 |
NA |
NA |
NA |
NA |
TTD |
| NTRK3 |
N-(1H-imidazol-5-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| NTSR1 |
2-(9H-fluoren-9-ylmethoxycarbonylamino)-4-methylpentanoic acid |
NA |
NA |
NA |
215500 |
NA |
NA |
BindingDB |
| NTSR1 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-6-[3-[3-[4-(3-aminopropylamino)butylamino]propylamino]propylamino]hexanoyl]amino]-6-aminohexanoyl]amino]-6-aminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NTSR1 |
(R)-4-methyl-2-(2-(5-(quinoline-8-sulfonamido)-1H-indol-1-yl)acetamido)pentanoic acid |
NA |
NA |
NA |
178000|178010 |
NA |
NA |
BindingDB |
| ODC1 |
N-delta-chloroacetyl-L-ornithine |
NA |
NA |
2500000 |
NA |
NA |
NA |
BindingDB |
| ODC1 |
Ornithine |
NA |
NA |
250000 |
NA |
NA |
NA |
BindingDB|PubChem |
| OGA |
N-[1-(7-aminoheptyl)-4,5-dihydroxy-6-(hydroxymethyl)piperidin-3-yl]acetamide, 2 |
107700 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OGA |
N-[4,5-dihydroxy-6-(hydroxymethyl)-1-(7-{[(4-methoxyphenyl)methyl]amino}heptyl)piperidin-3-yl]acetamide, 3 |
101500 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OGA |
N-[1-(7-{bis[(4-methoxyphenyl)methyl]amino}heptyl)-4,5-dihydroxy-6-(hydroxymethyl)piperidin-3-yl]acetamide, 4 |
175600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OGA |
N-{7-[5-acetamido-3,4-dihydroxy-2-(hydroxymethyl)piperidin-1-yl]heptyl}-5-{2-oxo-hexahydro-1H-thieno[3,4-d]imidazolidin-4-yl}pentanamide, 6 |
145000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OGA |
N-[1-(7-azidoheptyl)-4,5-dihydroxy-6-(hydroxymethyl)piperidin-3-yl]acetamide, 5 |
155100 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRD1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRD1 |
9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-1H-xanthene-1,8(2H)-dione |
NA |
NA |
NA |
141253754|190546072 |
NA |
NA |
BindingDB |
| OPRD1 |
Moxifloxacin |
NA |
NA |
NA |
NA |
NA |
299999 |
PubChem |
| OPRD1 |
3,3,6,6-tetramethyl-9-[4-[(2-propan-2-ylphenyl)methoxy]phenyl]-4,5,7,9-tetrahydro-2H-xanthene-1,8-dione |
NA |
NA |
NA |
204173794|354813389 |
NA |
NA |
BindingDB |
| OPRD1 |
9-[4-(cyclopentylmethoxy)phenyl]-3,3,6,6-tetramethyl-4,5,7,9-tetrahydro-2H-xanthene-1,8-dione |
NA |
NA |
NA |
27542287|275422870 |
NA |
NA |
BindingDB |
| OPRD1 |
9-[4-(cyclobutylmethoxy)phenyl]-3,3,6,6-tetramethyl-4,5,7,9-tetrahydro-2H-xanthene-1,8-dione |
NA |
NA |
NA |
34673685|346736850 |
NA |
NA |
BindingDB |