| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NT5E |
3-Fluoro-5-[6-(furan-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[4-Methoxy-6-(2-methylpyrazol-3-yl)benzotriazol-1-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(Furan-3-yl)imidazo[1,2-a]pyridin-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
2-Fluoro-3-[6-(furan-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
450000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(2-Methylpyrazol-3-yl)-4-pyrrolidin-1-ylbenzotriazol-1-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[5-(furan-3-yl)-1H-indazol-3-yl]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-[6-(1,2-Oxazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]phenol |
NA |
191000 |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
disodium;4-amino-1-[(2R,3R,4S,5S)-3,4-dihydroxy-5-[(1S)-1-hydroxy-2-phosphonatoethyl]oxolan-2-yl]pyrimidin-2-one |
1e+06|1000000 |
NA |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| NT5E |
Fludarabine |
5e+05|9e+05|500000|900000 |
NA |
NA |
NA |
NA |
NA |
ChEMBL|PubChem|TTD |
| NT5E |
Sodium anthraquinone-2,6-disulfonate |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| NT5E |
3-phenyl-N-(7H-purin-6-yl)benzamide |
893300|950000|1484100|2440300|3355700|6272500 |
NA |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| NTMT1 |
Allethrins |
NA |
NA |
NA |
NA |
141254 |
NA |
PubChem |
| NTMT1 |
4-Fluorofentanyl |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| NTMT1 |
Bexarotene |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| NTRK1 |
2-[(3R,4R)-3-fluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxy-4-(2-hydroxy-2-methylpropoxy)benzamide |
NA |
410000 |
NA |
NA |
NA |
NA |
TTD |
| NTRK1 |
Zabedosertib |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| NTRK1 |
Irak4-IN-20 |
NA |
636000 |
NA |
NA |
NA |
NA |
BindingDB |
| NTRK1 |
5-Methyl-3-(trifluoromethyl)indeno[2,1-b]quinoline-6,11-dione |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| NTRK1 |
7-Hydroxy-5-methylindeno[2,1-b]quinoline-6,11-dione |
NA |
141000 |
NA |
NA |
NA |
NA |
TTD |
| NTRK1 |
10-Methoxy-5-methylindeno[2,3-b]quinoline-6,11-dione |
NA |
209000 |
NA |
NA |
NA |
NA |
TTD |