| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| OPRD1 |
1-(1-cyclooctylpiperidin-4-yl)-3-[[(2S)-2,3-dihydroxypropyl]amino]quinoxalin-2-one |
530892 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRD1 |
2-[[4-(1-Cyclooctylpiperidin-4-yl)-3-oxoquinoxalin-2-yl]amino]acetamide |
548766 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRD1 |
4-[(1R,5S)-9-(1-adamantyl)-9-azabicyclo[3.3.1]nonan-3-yl]-3-oxoquinoxaline-2-carboxylic acid |
525570 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRD1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| OPRD1 |
4-[(1R,5S)-8-(1-adamantyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-oxoquinoxaline-2-carboxylic acid |
533800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRD1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRD1 |
8-[Bis(2-chlorophenyl)methyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one |
150385 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| OPRK1 |
(2R)-2-[(4S)-4-amino-8-hydroxy-3-oxo-4,5-dihydro-1H-2-benzazepin-2-yl]-N-[(4S)-2-(2-amino-2-oxoethyl)-3-oxo-4,5-dihydro-1H-2-benzazepin-4-yl]propanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRK1 |
(7S,12bS)-9-methoxy-7-[2-[2-[2-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-3-methyl-2,4,4a,7,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline |
108317.5 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRK1 |
(1R,2S,6R,14S)-11-methoxy-2-[2-[2-[2-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-N,N,14-trimethyl-15-oxatetracyclo[10.2.1.05,14.08,13]pentadeca-3,8(13),9,11-tetraen-6-amine |
108318 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRK1 |
H-Tyr-NMe-D-Ala-Phe-Sar-NH2 |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRK1 |
2-[5-[(3,4-Dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridine |
NA |
NA |
NA |
140000 |
NA |
NA |
BindingDB |
| OPRK1 |
(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol |
820000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| OPRK1 |
(2S)-2-amino-N-[(2R)-1-[[(4S)-2-(2-amino-2-oxoethyl)-3-oxo-4,5-dihydro-1H-2-benzazepin-4-yl]amino]-1-oxopropan-2-yl]-3-(4-hydroxy-2,6-dimethylphenyl)-N-methylpropanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRK1 |
(2S)-2-amino-N-[(2R)-1-[[(4S)-2-(2-amino-2-oxoethyl)-3-oxo-4,5-dihydro-1H-2-benzazepin-4-yl]amino]-1-oxopropan-2-yl]-3-(4-hydroxy-2,6-dimethylphenyl)propanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRK1 |
H-Tyr(2,6-diMe)-D-N(Me)Ala-Phe-Sar-NH2 |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRK1 |
(4R,4aR,6R,7S,7aR,12bS)-9-methoxy-3-methyl-2,4,4a,5,6,7,7a,13-octahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-6,7-diol |
NA |
NA |
NA |
126000 |
NA |
NA |
BindingDB|TTD |
| OPRM1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
Zilpaterol Hydrochloride |
130000|NA |
NA|320000|300000|1000000 |
NA |
NA |
NA |
NA |
PubChem |
| OPRM1 |
H-Tyr-DL-Pro-Leu-Asp-Leu-OH |
NA |
1085000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |