| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| OTC |
Medronic Acid |
9000000|20000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| OTC |
[Hydroxy(oxido)phosphoryl] phosphate |
240000|890000|2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OTC |
(2S)-2-ammonio-4-[({[(hydroxyphosphinato)methyl]phosphinato}methyl)ammonio]butanoate |
2300000|3200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OTC |
(2S)-2-[(tert-butoxycarbonyl)amino]-5-[({[(hydroxyphosphinato)methyl]phosphinato}methyl)ammonio]pentanoate |
1000000|2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OTC |
(Aminomethyl-hydroxy-phosphinoylmethyl)-phosphonic acid |
265000|800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OTC |
2-Amino-5-[(hydroxy-phosphonomethyl-phosphinoylmethyl)-amino]-pentanoic acid |
660000|750000|1900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX1 |
N-[3,5-bis(trifluoromethyl)phenyl]-2-chlorobenzamide |
NA |
539000 |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX1 |
N-[3,5-bis(trifluoromethyl)phenyl]-3-chloro-benzamide |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX4 |
2-Hydroxycarbamazepine |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| P2RX4 |
Basilen Blue |
NA |
NA |
NA |
128000 |
NA |
NA |
BindingDB |
| P2RX4 |
Reactive Blue-2 |
NA |
NA |
NA |
128000 |
NA |
NA |
TTD |
| P2RX7 |
N'-[2-chloro-4-(trifluoromethyl)phenyl]pentacyclo[6.4.0.02,10.03,7.04,9]dodeca-5,11-diene-8-carbohydrazide |
NA |
1557000 |
NA |
NA |
NA |
NA |
TTD |
| P2RX7 |
N'-(2-chlorophenyl)pentacyclo[6.4.0.02,10.03,7.04,9]dodecane-8-carbohydrazide |
NA |
933000 |
NA |
NA |
NA |
NA |
TTD |
| P2RX7 |
N'-[2-(trifluoromethyl)phenyl]pentacyclo[6.4.0.02,10.03,7.04,9]dodeca-5,11-diene-8-carbohydrazide |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| P2RX7 |
N'-[2-(trifluoromethyl)phenyl]pentacyclo[6.4.0.02,10.03,7.04,9]dodecane-8-carbohydrazide |
NA |
366000 |
NA |
NA |
NA |
NA |
TTD |
| P2RX7 |
2-[[4-(Furan-2-ylmethoxymethyl)triazol-1-yl]methyl]-3-methylnaphthalene-1,4-dione |
NA |
184400 |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX7 |
2-[[4-(Furan-2-ylmethoxymethyl)triazol-1-yl]-phenylmethyl]-3-methylnaphthalene-1,4-dione |
NA |
139600 |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX7 |
2-[[4-(Furan-2-ylmethoxymethyl)triazol-1-yl]-(4-nitrophenyl)methyl]-3-methylnaphthalene-1,4-dione |
NA |
183100 |
NA |
NA |
NA |
NA |
BindingDB |
| P2RX7 |
Adenosine Triphosphate |
NA |
NA |
NA |
780000 |
NA |
NA |
GtoPDB|PubChem|TTD |
| P2RY1 |
Hexasodium;8-[[4-fluoro-3-[[3-[[3-[[2-fluoro-5-[(4,6,8-trisulfonatonaphthalen-1-yl)carbamoyl]phenyl]carbamoyl]phenyl]carbamoylamino]benzoyl]amino]benzoyl]amino]naphthalene-1,3,5-trisulfonate |
NA |
1819700.86 |
NA |
NA |
NA |
NA |
TTD |