| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| OPRM1 |
H-Tyr-DL-Pro-Leu-Asp-Leu-Phe-OH |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| OPRM1 |
methyl (1R,9S,11S,15S,17S,19R)-19-(acetyloxymethyl)-14-ethylidene-18-oxa-2,12-diazahexacyclo[9.6.1.19,15.01,9.03,8.012,17]nonadeca-3,5,7-triene-19-carboxylate |
132000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| OPRM1 |
Zilpaterol |
130000 |
320000 |
NA |
NA |
NA |
NA |
BindingDB |
| OPRM1 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
(S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-methoxy-6-methylphenyl)methanone |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| OPRM1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| OPRM1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| OPRM1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| OPRM1 |
3-[(7R)-7-(cyclopropylmethylamino)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]nonan-5-yl]phenol |
NA |
NA |
NA |
130000 |
NA |
NA |
BindingDB|TTD |
| ORAI1 |
1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenoxyethanone |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| ORAI1 |
Diphenhydramine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| ORAI2 |
Diphenhydramine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| ORAI3 |
Diphenhydramine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| ORM1 |
(4R,5S)-2-{[(3S,4S,5S)-2-{[(2S,3S)-5-acetamido-6-hydroxy-2-(hydroxymethyl)-4-{[(2S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxy}oxan-3-yl]oxy}-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy}-4-hydroxy-5-[({2-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamido}carbonyl)amino]-6-[(1R,2R)-1,2,3-trihydroxypropyl]oxane-2-carboxylate |
NA |
8000000 |
NA |
NA |
NA |
NA |
BindingDB |
| ORM1 |
2-[2-(3,4,5-Trihydroxy-6-{[2-(1-phenyl-ethylcarbamoyl)-benzoylamino]-methyl}-tetrahydro-pyran-2-yl)-acetylamino]-pentanedioic acid |
NA |
5000000 |
NA |
NA |
NA |
NA |
BindingDB |
| OTC |
Phosphoric Acid |
6000000|12000000|20000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| OTC |
Pyrophosphoric acid |
240000|2000000|890000 |
NA |
NA |
NA |
NA |
NA |
PubChem |