| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PADI1 |
F-amidine |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
N-[(2S)-1-(benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]furan-2-carboxamide |
1086000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
Lucid-21-302 |
155000|402000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PADI1 |
US10716791, Code KP-305 |
147000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-310 |
3430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-313 |
1086000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-314 |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
N-[(2S)-1-(benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]-4-fluorobenzamide |
77690000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-288 |
353000|914000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
5,5-dimethyl-3-[2-(2H-tetrazol-5-yl)ethyl]imidazolidine-2,4-dione |
384000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
5,5-Dimethyl-3-[2-(2-methylimidazol-1-yl)ethyl]imidazolidine-2,4-dione |
2417000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
N-[(2S)-1-(benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]-1-methylpyrrole-2-carboxamide |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-286 |
964000|2495000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-298 |
785000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
US10716791, Code KP-303 |
392000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
2-chloro-N'-[3-[5-chloro-4-(3-phenylphenyl)-1H-imidazol-2-yl]propyl]ethanimidamide |
NA |
161000 |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
(E)-4-[(1-amino-2-chloroethylidene)amino]-N-[(3-phenylphenyl)methyl]but-2-enamide |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
2-chloro-N'-[3-[1-(3-phenylphenyl)triazol-4-yl]propyl]ethanimidamide |
NA |
294000 |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
4-[(1-amino-2-chloroethylidene)amino]-N-[(3-phenylphenyl)methyl]but-2-ynamide |
NA |
408000 |
NA |
NA |
NA |
NA |
BindingDB |
| PADI1 |
5,5-Dimethyl-3-(2-morpholin-4-ylethyl)imidazolidine-2,4-dione |
602000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |