Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PADI1 5,5-Dimethyl-3-(piperazin-1-ylmethyl)imidazolidine-2,4-dione 445000 NA NA NA NA NA BindingDB
PADI2 2-[(1-amino-2-chloroethylidene)amino]ethyl N-[(3-phenylphenyl)methyl]carbamate NA 151000 NA NA NA NA BindingDB
PADI2 1-[2-[(1-Amino-2-chloroethylidene)amino]ethyl]-3-[(3-phenylphenyl)methyl]urea NA 140000 NA NA NA NA BindingDB
PADI2 2-chloro-N'-[3-[1-(3-phenylphenyl)triazol-4-yl]propyl]ethanimidamide NA 110000 NA NA NA NA BindingDB
PADI2 4-[(1-amino-2-chloroethylidene)amino]-N-[(3-phenylphenyl)methyl]but-2-ynamide NA 153000 NA NA NA NA BindingDB
PADI3 F-amidine NA|293000 367000|NA NA NA NA NA BindingDB|TTD
PADI4 F-amidine 330000 NA NA NA NA NA BindingDB
PADI4 US10716791, Code KP-289 488000 NA NA NA NA NA BindingDB|TTD
PADI4 N-[(2S)-1-(benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]furan-2-carboxamide 2823000 NA NA NA NA NA BindingDB|TTD
PADI4 N-[(2S)-4-(4-methylpiperazin-1-yl)-1-oxo-1-(propan-2-ylamino)butan-2-yl]cyclohexanecarboxamide 10000000 NA NA NA NA NA TTD
PADI4 N-[(2S)-1-(benzylamino)-4-imidazol-1-yl-1-oxobutan-2-yl]furan-2-carboxamide 10000000 NA NA NA NA NA TTD
PADI4 US10716791, Code KP-287 10000000 NA NA NA NA NA TTD
PADI4 Lucid-21-302 180000 NA NA NA NA NA BindingDB|PubChem|TTD
PADI4 US10716791, Code KP-310 1453000 NA NA NA NA NA BindingDB
PADI4 US10716791, Code KP-313 2823000 NA NA NA NA NA BindingDB
PADI4 US10716791, Code KP-288 591000 NA NA NA NA NA BindingDB|TTD
PADI4 Methotrexate NA 10000000 NA NA NA NA PubChem|TTD
PADI4 US10716791, Code KP-286 714000 NA NA NA NA NA BindingDB
PADI4 2-chloro-N'-[3-(1-methylindol-3-yl)propyl]ethanimidamide NA 190000 NA NA NA NA BindingDB|TTD
PADI4 US10716791, Code KP-298 1238000 NA NA NA NA NA BindingDB