| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PADI4 |
US10716791, Code KP-300 |
1068000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
US10716791, Code KP-303 |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
US10716791, Code KP-292 |
14940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
1-[2-[(1-Amino-2-chloroethylidene)amino]ethyl]-3-[(3-phenylphenyl)methyl]urea |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
Streptomycin |
560000|NA |
NA|1800000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
Azathioprine |
NA |
8100000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PADI4 |
Cl-amidine |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
5,5-Dimethyl-3-(2-morpholin-4-ylethyl)imidazolidine-2,4-dione |
1430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
2-Fluoroethanimidamide |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
Leflunomide |
NA |
2400000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PADI4 |
Mesalamine |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
Clindamycin |
NA |
5100000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
Azithromycin |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
5,5-Dimethyl-3-(2-pyrrolidin-1-ylethyl)imidazolidine-2,4-dione |
4643000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
3-(2-Imidazol-1-ylethyl)-5,5-dimethylimidazolidine-2,4-dione |
632000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
Sulfamethoxazole |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
Sulfapyridine |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
(2E,4S,4aS,5aS,6S,12aS)-2-[azanyl(oxidanyl)methylidene]-4-(dimethylamino)-6-methyl-6,10,11,12a-tetrakis(oxidanyl)-4,4a,5,5a-tetrahydrotetracene-1,3,12-trione |
NA |
780000 |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
(2Z,4S,4aR,5S,5aR,6R,12aS)-2-[amino(hydroxy)methylene]-4-(dimethylamino)-5,10,11,12a-tetrahydroxy-6-methyl-4a,5,5a,6-tetrahydro-4H-tetracene-1,3,12-trione;ethanol;hydrate;hydrochloride |
NA|630000 |
860000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
CID 54575046 |
NA|180000|540000 |
620000|NA |
NA |
NA |
NA |
NA |
BindingDB |