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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PAM 2-[(2S)-2-amino-3-phenylpropanoyl]oxyacetic acid NA 1100000|1600000 NA NA NA NA BindingDB
PAM 2-[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carbonyl]oxyacetic acid NA 290000|370000 NA NA NA NA BindingDB
PAM 2-[(2S)-2-[[(2S)-2-[(2-aminoacetyl)amino]propanoyl]amino]-3-phenylpropanoyl]oxyacetic acid NA 160000|560000 NA NA NA NA BindingDB
PAM 2-[2-[[(2S)-2-acetamido-4-methylpentanoyl]amino]acetyl]oxyacetic acid NA 120000|200000 NA NA NA NA BindingDB
PAM 2-[(2S)-pyrrolidine-2-carbonyl]oxyacetic acid NA 500000|600000 NA NA NA NA BindingDB
PAM 2-[(2S)-1-[(2S)-2-[(2-aminoacetyl)amino]propanoyl]pyrrolidine-2-carbonyl]oxyacetic acid NA 980000|1100000 NA NA NA NA BindingDB
PAM 2-[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-phenylpropanoyl]oxyacetic acid NA 350000|370000 NA NA NA NA BindingDB
PAM 2-(2-Acetamidoacetoxy)Acetic Acid NA 210000|1800000 NA NA NA NA BindingDB
PAM Ac-Pro-OLeu-Gly-OGly-OH NA 180000 NA NA NA NA BindingDB
PAM Acetoxyacetic acid NA 1100000 NA NA NA NA BindingDB
PANX1 Probenecid NA 150000 NA NA NA NA PubChem
PAOX N-Acetylputrescine 800000 NA NA NA NA NA PubChem|TTD
PAOX 3-N-[(2-phenoxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX C3-Amide-C4-NH2 29000000 NA NA NA NA NA TTD
PAOX N-(6-aminohexyl)methanesulfonamide 376000 NA NA NA NA NA TTD
PAOX N-(8-aminooctyl)methanesulfonamide 650000 NA NA NA NA NA TTD
PAOX methyl N-(8-aminooctyl)carbamate 260000 NA NA NA NA NA TTD
PAOX N-(6-aminohexyl)-2-chloroacetamide 130000 NA NA NA NA NA TTD
PAOX 3-N-[(2-naphthalen-2-yloxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(5-methyl-2-propan-2-ylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD