| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PARG |
Benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PARG |
3,5-Dichloro-N-(3-chlorophenyl)-2-hydroxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PARG |
N,1,3-triethyl-2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-sulfonamide |
NA |
NA |
NA |
140000 |
NA |
NA |
TTD |
| PARG |
N-(tert-butyl)-2-oxo-1,2-dihydroquinoline-6-sulfonamide |
NA |
NA |
NA |
110000 |
NA |
NA |
TTD |
| PARG |
3,5-dichloro-N-(3-chloro-4-naphthalen-2-yloxyphenyl)-2-hydroxy-N-methylbenzamide |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| PARG |
N-(3-chloro-4-naphthalen-2-yloxyphenyl)-2-hydroxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PARG |
5-chloro-N-(3-chloro-4-naphthalen-2-yloxyphenyl)-2-hydroxybenzamide |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| PARG |
N-(2-hydroxyethyl)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PARG |
N-(2-methoxyethyl)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PARG |
N-tert-butylnaphthalene-2-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PARN |
1-hydroxy-7-(pyridin-2-ylmethyl)-3H-purine-2,6-dione |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
| PARN |
1-hydroxy-7-(pyridin-3-ylmethyl)-3H-purine-2,6-dione |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| PARN |
1-hydroxy-7-(pyridin-4-ylmethyl)-3H-purine-2,6-dione |
NA |
245000 |
NA |
NA |
NA |
NA |
BindingDB |
| PARN |
Nucleoside, A2 |
510000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PARN |
Nucleoside, A6 |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PARN |
Nucleoside, C6 |
645000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PARP1 |
Veliparib |
NA |
133500|NA |
NA |
NA|160000 |
NA |
NA |
PubChem |
| PARP1 |
4-Chlorobenzamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
1-(cyclopropylmethyl)-N-(1-methylcyclopropyl)-3-[(2-methyl-1,3-thiazol-5-yl)methyl]-2,4-dioxoquinazoline-6-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PARP1 |
1-(cyclopropylmethyl)-3-methyl-N-(1-methylcyclopropyl)-2,4-dioxoquinazoline-6-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |