| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PARP1 |
1-[(2,5-dimethylpyrazol-3-yl)methyl]-N-(1-methylcyclopropyl)-3-[(1-methylpyrazol-4-yl)methyl]-2,4-dioxoquinazoline-6-sulfonamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PARP1 |
3-Nitrobenzamide |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
5-fluoro-2-[(2R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide |
NA |
338000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
(3s,6s)-3,6-Dimethylpiperazine-2,5-dione |
NA |
900000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
3-(Dimethylamino)benzamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
3,5-Dichloro-N-(3-chlorophenyl)-2-hydroxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
3,5-dichloro-N-(3-chloro-4-naphthalen-2-yloxyphenyl)-2-hydroxybenzamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
3,5-dichloro-N-(2-chlorophenyl)-2-hydroxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
N-[4-(3-bromonaphthalen-2-yl)oxy-3-chlorophenyl]-3,5-dichloro-2-hydroxybenzamide |
NA |
123000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
4-Hydroxybenzamide |
NA |
280000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
(3R,6S)-3,6-dimethylpiperazine-2,5-dione |
NA |
4200000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
5'-O-[(S)-{[(S)-{[(2R,3R,4S)-3,4-Dihydroxypyrrolidin-2-YL]methoxy}(hydroxy)phosphoryl]oxy}(hydroxy)phosphoryl]adenosine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
4-Bromobenzamide |
NA |
2200000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
4-Fluorobenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
4-[[3-(2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-triene-2-carbonyl)-4-fluorophenyl]methyl]-2H-phthalazin-1-one |
NA |
156000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
6-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]-2,6-diazatricyclo[7.3.1.05,13]trideca-1(12),9(13),10-trien-3-one |
NA |
387000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
N-(1-oxo-3,4-dihydro-2H-isoquinolin-4-yl)-3-[(4-oxo-3H-phthalazin-1-yl)methyl]benzamide |
NA |
145750 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
4-Aminobenzamide |
NA |
1800000 |
NA |
NA |
NA |
NA |
TTD |
| PARP1 |
Niacinamide |
NA |
210000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PARP2 |
(4s)-3-{trans-4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]cyclohexyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |