| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PARP2 |
N-[4-[(4S)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-7-fluoro-1,5-naphthyridine-4-carboxamide |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| PARP2 |
1-[4-[(4S)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]-4-fluoro-2-oxo-3H-benzimidazole-5-carbonitrile |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| PARP2 |
(4s)-3-{4-[6-Amino-5-(Pyrimidin-2-Yl)pyridin-3-Yl]phenyl}-5,5-Dimethyl-4-Phenyl-1,3-Oxazolidin-2-One |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| PARP2 |
2-amino-5-[4-[(4S)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]cyclohexyl]pyridine-3-carbonitrile |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| PBRM1 |
3-Acetylindole |
NA |
NA |
1195000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
5-Chloro-2-(3-methylphenyl)-3,1-benzoxazin-4-one |
NA |
236000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
2-[(2-Chloro-6-fluorophenyl)methylideneamino]benzamide |
NA |
119000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
Methanone, (3-aminophenyl)phenyl- |
NA |
NA |
709000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
2,4-Di(3-pyridyl)-1,3-thiazole |
NA |
NA |
1387000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
5-Methyl-6-(2-thienyl)-2,3,4,5-tetrahydropyridazin-3-one |
NA |
NA |
1210000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
2-(2-chloro-6-fluorophenyl)-2,3-dihydro-1H-quinazolin-4-one |
NA |
NA |
179000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
4-Carboxy-9-acridanone |
NA |
127000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
5-(2-Bromophenyl)-1H-tetrazole |
NA |
NA |
1446000 |
NA |
NA |
NA |
ChEMBL |
| PBRM1 |
6-Hydroxy-1-indanone |
NA |
NA |
902000 |
NA |
NA |
NA |
ChEMBL |
| PCMT1 |
(2S,5R)-2,5-diamino-6-[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]hexanoic acid |
236000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PCMT1 |
Ademetionine |
164000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PCMT1 |
(2S)-2,5-diamino-6-[(2R,3S,4R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]hexanoic acid |
1680000|2500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PCMT1 |
Sinefungin |
126000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PCSK9 |
Benzeneboronic acid |
470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDCL3 |
ethyl 2-(4-oxo-4,5,6,7-tetrahydro-3H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-3-yl)acetate |
NA |
NA |
227000 |
NA |
NA |
NA |
BindingDB |