| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE10A |
5-Nitroquinoline |
590000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
2-Amino-4,6-dimethylpyrimidine |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
2-Methyl-4(3H)-quinazolinone |
990000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
4-Hydroxyquinazoline |
910000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
4-Amino-6-mercaptopyrazolo[3,4-d]pyrimidine |
450000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
3-Methyl-2-phenylquinoline |
NA |
NA |
424000 |
NA |
NA |
NA |
BindingDB |
| PDE10A |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
9-(2-ethylhexyl)-2-[(4-phenylmethoxyphenyl)methyl]-4,5-dihydro-1H-purin-6-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
9-(2-ethylhexyl)-2-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-purin-6-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDE10A |
|
990000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE10A |
6,7-dimethoxy-4-[(3R)-3-(naphthalen-1-yloxy)pyrrolidin-1-yl]quinazoline |
208000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE10A |
2-[(1-hydroxy-3H-2,1-benzoxaborol-5-yl)oxy]-6-(trifluoromethyl)quinoline |
NA |
4520000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE10A |
6,7-Dimethoxy-4-[4-(quinoxalin-2-ylmethyl)piperazin-1-yl]quinazoline |
NA |
169824 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE10A |
4-[3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)pyrrolidin-1-yl]-6,7-dimethoxyquinazoline |
NA |
104713 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE10A |
2h-Isoindole-1,3-Diamine |
380000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
2-(4-Methyl-2-thiazolyl)pyridine |
NA |
324000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
5-Nitroindazole |
560000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
2-Amino-4-methyl-3-nitropyridine |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE10A |
2,3-Dihydro-1,4-benzodioxin-6-methanol |
940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |