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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PDE10A 2,3-Dimethylquinoline-4-carboxylic acid NA NA 505000 NA NA NA BindingDB
PDE10A 2-Benzothiazolamine, 4-chloro- 210000 NA NA NA NA NA BindingDB|TTD
PDE10A Crisaborole NA 97600000 NA NA NA NA BindingDB|PubChem
PDE10A Roflumilast NA 200000 NA NA NA NA PubChem
PDE10A Rolipram NA 140000 NA NA NA NA BindingDB|PubChem
PDE10A 2-[3-[3-(1-Methylsulfonylpiperidin-4-yl)pyrazin-2-yl]oxyazetidin-1-yl]quinoline NA 166000 NA NA NA NA BindingDB|TTD
PDE10A 2-[3-[3-[4-(Methoxymethyl)piperidin-1-yl]pyrazin-2-yl]oxyazetidin-1-yl]quinoline NA 147000 NA NA NA NA BindingDB|TTD
PDE10A 2-[3-(3-Pyridin-2-ylpyrazin-2-yl)oxyazetidin-1-yl]quinoline NA 350000 NA NA NA NA BindingDB|TTD
PDE10A N,N-dimethyl-1-[3-(1-quinolin-2-ylazetidin-3-yl)oxypyrazin-2-yl]piperidin-4-amine NA 343000 NA NA NA NA BindingDB|TTD
PDE10A 2-[3-[3-(4-Methylphenyl)pyrazin-2-yl]oxyazetidin-1-yl]quinoline NA 107000 NA NA NA NA BindingDB|TTD
PDE10A 2-[3-(3-Pyrimidin-5-ylpyrazin-2-yl)oxyazetidin-1-yl]quinoline NA 125000 NA NA NA NA BindingDB|TTD
PDE10A 2-[3-[3-(4-Methylpiperidin-1-yl)pyrazin-2-yl]oxyazetidin-1-yl]quinoline NA 103000 NA NA NA NA BindingDB|TTD
PDE10A 910000 NA NA NA NA NA BindingDB
PDE10A 7-Chloro-4-hydroxyquinoline 500000 NA NA NA NA NA BindingDB|TTD
PDE10A 2,4-Diamino-6-chloropyrimidine 410000 NA NA NA NA NA BindingDB|TTD
PDE10A 5-(2-Furyl)-3-methyl-1H-pyrazole NA 851000 NA NA NA NA BindingDB|TTD
PDE10A 5-Nitrobenzimidazole 500000 NA NA NA NA NA BindingDB|PubChem|TTD
PDE10A 6-chloro-3-[(dimethylamino)methyl]-2-phenyl-1H-quinolin-4-one NA NA 102000 NA NA NA BindingDB
PDE10A 1,4-Benzodioxan-6-yl methyl ketone 1200000 NA NA NA NA NA BindingDB|TTD
PDE10A Cinchophen NA NA 127000 NA NA NA BindingDB|PubChem