| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE10A |
2-[4-Fluoro-3-[7-methyl-12-(trifluoromethyl)-2,4,5,8,13-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-3-yl]phenyl]propan-2-ol |
NA |
7980000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE11A |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE11A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE11A |
Rolipram |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE11A |
Zardaverine |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1A |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE1A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE1A |
Theophylline |
NA |
320000|356000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Cilostazol |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Amrinone |
NA |
1000000|300000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Milrinone |
NA |
340000|198000|310000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Crisaborole |
NA |
5600000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Rolipram |
NA|200000 |
200000|NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE1A |
Enoximone |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE1B |
MS 857 |
NA |
409000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1B |
6-(4-(1H-Imidazol-1-yl)phenyl)pyridazin-3-ol |
NA |
580000|660000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1B |
4,5-dihydro-6-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinone |
NA |
530000|790000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1B |
6-[4-(1H-Imidazol-2-yl)-phenyl]-2H-pyridazin-3-one |
NA |
330000|460000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1B |
6-(4-Benzoimidazol-1-yl-phenyl)-4,5-dihydro-2H-pyridazin-3-one |
NA |
220000|280000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE1B |
4,5-Dihydro-6-[4-(4,5,6,7-tetrahydro-1H-benzimidazol-1-yl)phenyl]-3(2H)-pyridazinone |
NA |
140000|180000 |
NA |
NA |
NA |
NA |
BindingDB |