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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PDE1C Cilostazol NA 1000000 NA NA NA NA PubChem
PDE1C Amrinone NA 300000|1000000 NA NA NA NA PubChem
PDE1C Milrinone NA 310000|198000|340000 NA NA NA NA PubChem
PDE1C Crisaborole NA 71000000 NA NA NA NA PubChem
PDE1C Rolipram 200000|NA NA|200000 NA NA NA NA PubChem
PDE1C Enoximone NA 1000000 NA NA NA NA PubChem
PDE2A Tadalafil NA 130000 NA NA NA NA BindingDB|PubChem
PDE2A 9-(2-fluorobenzyl)-6-(methylamino)-9H-purine 122000 NA NA NA NA NA TTD
PDE2A 6-(4-(1H-Imidazol-1-yl)phenyl)pyridazin-3-ol NA 190000 NA NA NA NA TTD
PDE2A 6-(4-Imidazol-1-yl-phenyl)-2-methyl-4,5-dihydro-2H-pyridazin-3-one NA 280000 NA NA NA NA TTD
PDE2A 6-(4-Imidazol-1-yl-phenyl)-4-methyl-4,5-dihydro-2H-pyridazin-3-one NA 260000 NA NA NA NA TTD
PDE2A 4,5-dihydro-6-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinone NA 380000 NA NA NA NA TTD
PDE2A 6-[4-(1H-Imidazol-2-yl)-phenyl]-2H-pyridazin-3-one NA 190000 NA NA NA NA TTD
PDE2A 4,5-dihydro-6-[4-(4-hydroxymethyl-1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinone NA 480000 NA NA NA NA TTD
PDE2A 6-(3-Imidazol-1-yl-phenyl)-4,5-dihydro-2H-pyridazin-3-one NA 330000 NA NA NA NA TTD
PDE2A 6-(4-(1H-Imidazol-1-yl)phenyl)-5-methylpyridazin-3(2H)-one NA 170000 NA NA NA NA TTD
PDE2A 4-amino-6-(4-imidazol-1-ylphenyl)-2H-pyridazin-3-one NA 110000 NA NA NA NA TTD
PDE2A 2-[6-Fluoro-8-methylsulfonyl-9-[[4-(trifluoromethyl)phenyl]methyl]-1,2,3,4-tetrahydrocarbazol-1-yl]acetonitrile NA 278000 NA NA NA NA TTD
PDE2A Cilomilast NA 160000 NA NA NA NA BindingDB|PubChem
PDE2A 6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide NA 200000 NA NA NA NA TTD