| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE2A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
8-Methoxymethyl-3-isobutyl-1-methylxanthine |
NA |
212000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
1H-Purine-2,6-dione, 3,7-dihydro-7-(2-hydroxypropyl)-1,3-dimethyl-, (S)- |
700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
1H-Purine-2,6-dione, 3,7-dihydro-7-(2-hydroxypropyl)-1,3-dimethyl-, (R)- |
600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
4,5-dihydro-6-[4-(2-ethyl-4-methyl-1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinone |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
Theophylline |
NA |
210000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE2A |
4,5-dihydro-6-(4-(imidazol-1-yl)phenyl)-5-methyl-3(2H)-pyridazinone |
NA |
380000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
1H-Purine-2,6-dione, 3,7-dihydro-1-methyl-3-(2-methylpropyl)-7-(phenylmethyl)- |
NA |
108000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
Amrinone |
NA |
580000|700000|720000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE2A |
Milrinone |
NA |
220000|200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE2A |
4-(4-Imidazol-1-yl-phenyl)-4a,5,6,7,8,8a-hexahydro-2H-phthalazin-1-one |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
Crisaborole |
NA |
3630000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE2A |
Roflumilast |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE2A |
Proxyphylline |
600000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE2A |
4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone |
NA |
390000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
Rolipram |
NA|200000 |
200000|NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE2A |
Sulmazole |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE2A |
Enoximone |
NA |
520000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE2A |
Imazodan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-[3-(dimethylamino)-2-hydroxypropoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |