| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE3A |
2-[2-(8-Chloro-2-oxospiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-5-yl)oxyethylamino]acetic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE3A |
2-butyl-N-[(4-phenylphenyl)methyl]thieno[3,2-d]pyrimidin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
(1-Methylbenzimidazol-2-yl)-[4-(3-pyridin-3-ylpyridin-2-yl)oxyphenyl]methanone |
NA |
167000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
5-Benzyl-2-pentylpyrazolo[4,3-c]quinolin-3-one |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
5-Benzyl-2-(cyclohexylmethyl)pyrazolo[4,3-c]quinolin-3-one |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4-Fluoro-2-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
199000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
4-[2-[2-(2-Fluoroethoxy)ethoxy]ethoxy]-2-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
4-[2-[2-[2-(2-Fluoroethoxy)ethoxy]ethoxy]ethoxy]-2-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
144400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
4-(2-Fluoroethoxymethyl)-2-[[4-(2-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
306000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
6-Fluoro-2-[[4-(2-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
6-[4-(2-ethoxy-2-phenylethyl)piperazin-1-yl]sulfonyl-N-methyl-N-phenylquinazolin-4-amine |
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2-oxo-5-pyridin-4-yl-1H-pyridine-3-carbonitrile |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
6-(4-Imidazol-1-yl-phenyl)-2-methyl-4,5-dihydro-2H-pyridazin-3-one |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
3-(3-methyl-2-phenylimidazol-4-yl)-1H-pyridazin-6-one |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
3-[2-(3,4-dimethoxyphenyl)-1-methylimidazol-4-yl]-4,5-dihydro-1H-pyridazin-6-one |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4-methyl-6-(4-methylpiperazin-1-yl)-3H-quinazolin-2-one |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2,4,7,13-Tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,10,12-tetraen-5-one |
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
5,8-dimethoxy-4-methyl-3H-quinazolin-2-one |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
6,8-dimethoxy-4-methyl-3H-quinazolin-2-one |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |