| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE3A |
ethyl 2-methyl-6-oxo-5-propyl-1H-pyridine-3-carboxylate |
NA |
125100 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
7,8-dimethoxy-N-[1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]quinazolin-4-amine |
NA |
101000|369000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
(11R,15S)-4-ethyl-8-methyl-1,3,5,8,10-pentazatetracyclo[7.6.0.02,6.011,15]pentadeca-2(6),3,9-trien-7-one |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
(11R,15S)-8-methyl-4-pentan-3-yl-1,3,5,8,10-pentazatetracyclo[7.6.0.02,6.011,15]pentadeca-2(6),3,9-trien-7-one |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4-(4-Imidazol-1-yl-phenyl)-4a,5,6,7,8,8a-hexahydro-2H-phthalazin-1-one |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2-Butyl-5-(cyclohexylmethyl)pyrazolo[4,3-c]quinolin-3-one |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2-butyl-1H-pyrazolo[4,3-c]quinolin-3-one |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
6-(4-Methylsulfonyl-2,3-dihydro-1,4-benzoxazin-6-yl)-2-phenyl-4,5-dihydropyridazin-3-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
N-ethyl-N-[[4-[2-(tetrazol-2-yl)phenyl]phenyl]methyl]-[1,2,4]thiadiazolo[2,3-a]benzimidazol-2-amine |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
Crisaborole |
NA |
64000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE3A |
Proxyphylline |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE3A |
Rolipram |
NA|200000 |
242000|NA|300000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE3A |
Sulmazole |
NA |
150000|500000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-methylpyridazin-3(2H)-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-3-yl)-4,5-dihydropyridazin-3(2H)-one |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
2-benzyl-6-(2-isopropyl-7-methoxypyrazolo[1,5-a]pyridin-3-yl)-4,5-dihydropyridazin-3(2H)-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
15-Propan-2-yl-3,4,13,14-tetrazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,9,11,14-pentaen-5-one |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
3-(6-Chloro-4-methylpyridazin-3-yl)-2-isopropylpyrazolo[1,5-a]pyridine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
2-Isopropyl-3-(6-methoxypyridazin-3-yl)pyrazolo[1,5-a]pyridine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
(S)-6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-methyl-4,5-dihydropyridazin-3(2H)-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |