| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE3A |
6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-4,5-dihydropyridazin-3(2H)-one |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
2-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-phenol |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-[2-(methylamino)ethoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-(4-fluoro-phenyl)-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
5-(2-Aminoethoxy)-8-chlorospiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-[2-hydroxy-3-(methylamino)propoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-(3-fluoro-phenyl)-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-[2-(dimethylamino)ethoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-[3-(dimethylamino)propoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
5-[2-(2-Aminoethoxy)ethoxy]-8-chlorospiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3B |
Tadalafil |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE3B |
(1-Methylbenzimidazol-2-yl)-[4-(3-pyridin-3-ylpyridin-2-yl)oxyphenyl]methanone |
NA |
234000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3B |
4-Fluoro-2-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3B |
4-(2-Fluoroethoxymethyl)-2-[[4-(2-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3B |
6-Fluoro-2-[[4-(2-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
151000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3B |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3B |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3B |
2-[(1-hydroxy-3H-2,1-benzoxaborol-5-yl)oxy]-6-(trifluoromethyl)quinoline |
NA |
7190000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3B |
Theophylline |
NA |
240000|360000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE3B |
Amrinone |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |