Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| PDE3B | Crisaborole | NA | 58800000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE3B | Roflumilast | NA | 200000 | NA | NA | NA | NA | PubChem |
| PDE3B | Proxyphylline | 1000000 | NA | NA | NA | NA | NA | PubChem |
| PDE3B | Rolipram | NA|200000 | 300000|242000|NA|200000 | NA | NA | NA | NA | PubChem |
| PDE4A | Xanthine | 200000 | NA | NA | NA | NA | NA | PubChem |
| PDE4A | Theophylline | NA | 386000|1780000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE4A | Caffeine | NA | 747000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE4A | Amrinone | NA | 150000|126000|101000 | NA | NA | NA | NA | PubChem |
| PDE4A | Pentoxifylline | NA | 168000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| PDE4A | 4-imino-7-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-3(4H)-amine | NA|153000 | 757000|1760000|NA | NA | NA | NA | NA | BindingDB |
| PDE4A | Enoximone | NA | 150000 | NA | NA | NA | NA | PubChem |
| PDE4A | Thalidomide | NA | 500000 | NA | NA | NA | NA | PubChem |
| PDE4A | diaminomethylidene-[(Z)-1-(3,3-dimethylcyclohexen-1-yl)ethylideneamino]azanium | NA|127000 | 790000|1460000|NA | NA | NA | NA | NA | BindingDB |
| PDE4A | 5,5-Dimethyl-3-(piperazin-1-ylmethyl)imidazolidine-2,4-dione | NA|131000|371000 | 1380000|4269000|NA | NA | NA | NA | NA | BindingDB|TTD |
| PDE4A | 3-Methylxanthine | 156000 | NA | NA | NA | NA | NA | PubChem |
| PDE4A | N-[4-[(3R)-2,3-Dihydro-3-methyl-2-oxo-1H-indol-5-yl]-2-thiazolyl]guanidine | NA|115000|231000 | 1320000|2650000|NA | NA | NA | NA | NA | BindingDB|TTD |
| PDE4A | 3-Methoxy-2-[[4-(2-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline | NA | 199000 | NA | NA | NA | NA | BindingDB|TTD |
| PDE4B | HC-030031 | NA | 200000 | NA | NA | NA | NA | TTD |
| PDE4B | Xanthine | 200000 | NA | NA | NA | NA | NA | PubChem |
| PDE4B | 4-[8-(benzylamino)-1,3-dimethyl-2,6-dioxopurin-7-yl]-N-[(E)-(2-hydroxyphenyl)methylideneamino]butanamide | NA | 200000 | NA | NA | NA | NA | TTD |