| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE4B |
ethyl 1-[3,5-bis(trifluoromethyl)phenyl]-3,5-dimethyl-1H-pyrazole-4-carboxylate |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE4B |
6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)pyridazin-3(2H)-one |
NA |
114000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4B |
Amrinone |
NA |
126000|101000|150000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4B |
Enoximone |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4B |
Thalidomide |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4B |
6-(2-isopropylpyrazolo[1,5-a]pyridin-3-yl)-5-methylpyridazin-3(2H)-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4B |
3,4,11,12-Tetrazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(17),2,10,13,15-pentaen-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4B |
3-(6-Chloro-4-methylpyridazin-3-yl)-2-isopropylpyrazolo[1,5-a]pyridine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4B |
2-Isopropyl-3-(6-methoxypyridazin-3-yl)pyrazolo[1,5-a]pyridine |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4B |
3-Methylxanthine |
156000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
Xanthine |
200000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
Theophylline |
NA |
1780000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
Amrinone |
NA |
101000|126000|150000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
Enoximone |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
Thalidomide |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4C |
3-Methylxanthine |
156000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
Xanthine |
200000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
2-(4-chlorophenyl)sulfonyl-7-cyclopentyloxy-6-methoxy-3,4-dihydro-1H-isoquinoline |
NA |
133560 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
Theophylline |
NA |
1780000 |
NA |
NA |
NA |
NA |
PubChem |