| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE4D |
3-Methylxanthine |
156000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
N-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-cyclohexane-1,4-diamine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
2-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-phenol |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-(4-fluoro-phenyl)-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
3-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-phenol |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-(3-fluoro-phenyl)-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
N-(2-bicyclo[2.2.1]heptanyl)-5-(4-chlorophenyl)-3-methyl-1,3,4-thiadiazol-2-imine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
4-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-benzoic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
N-(4-Chloro-phenyl)-3-cyclopentyloxy-4-methoxy-benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
N-(2-chloro-6-methyl-phenyl)-3-cyclopentyloxy-4-methoxy-benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
3-(cyclopentyloxy)-N-(2-fluorophenyl)-4-methoxybenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
3-Cyclopentyloxy-N-(2,5-dichloro-phenyl)-4-methoxy-benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
8-Chloro-5-[3-(dimethylamino)-2-hydroxypropoxy]spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
5-[(8-Chloro-2-oxospiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-5-yl)oxymethyl]furan-2-carboxylic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
N-(2-chloro-6-fluoro-phenyl)-3-cyclopentyloxy-4-methoxy-benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
3-(cyclopentyloxy)-N-(2,6-dichlorophenyl)-4-methoxybenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
2-[2-(8-Chloro-2-oxospiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-5-yl)oxyethylamino]acetic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
3-cyclopentyloxy-4-methoxy-N-(2-methylsulfanylphenyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE5A |
3-Cyclopentyloxy-4-methoxy-N-(2-trifluoromethyl-phenyl)-benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |