| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE4D |
{1-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-cyclopentyl}-methanol |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
[5-(3-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-cyclohexyl-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
4-{5-[(Z)-Cyclohexylimino]-4-methyl-4,5-dihydro-[1,3,4]thiadiazol-2-yl}-2-methoxy-benzamide |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
4-{5-[(Z)-Cyclohexylimino]-4-methyl-4,5-dihydro-[1,3,4]thiadiazol-2-yl}-N-(2-dimethylamino-ethyl)-N-methyl-benzamide |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylidene]-(1-ethyl-propyl)-amine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
1-[4-Methoxy-3-(piperidin-4-yloxy)phenyl]pentan-1-one |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
1-[3-Methoxy-4-(tetrahydropyran-4-yloxy)phenyl]butan-1-ol |
NA |
1513561.25 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
1-[3-Methoxy-4-(tetrahydropyran-4-yloxy)phenyl]pentan-1-ol |
NA |
537031.8 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
1-[3-Methoxy-4-(tetrahydrofuran-3-yloxy)phenyl]butan-1-ol |
NA |
524807.46 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
Amrinone |
NA |
101000|150000|126000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
5-(4-chlorophenyl)-N-cyclooctyl-3-methyl-1,3,4-thiadiazol-2-imine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE4D |
Enoximone |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
Thalidomide |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE4D |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE4D |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| PDE4D |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| PDE4D |
7-{5-[(Z)-Cyclohexylimino]-4-methyl-4,5-dihydro-[1,3,4]thiadiazol-2-yl}-quinazolin-4-ylamine |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |