| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE3A |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE3A |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE3A |
|
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
(5-Phenylfuran-2-yl)methyl 3,4,5-triethoxybenzoate |
NA |
104200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| PDE3A |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| PDE3A |
6-Methoxy-1-methylisoquinolin-3(2H)-one |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
8-Chloro-6-phenylspiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
8-Chloro-5-(2-morpholin-4-ylethoxy)spiro[1,3-dihydroquinazoline-4,1'-cyclohexane]-2-one |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
ethyl 5-[(3-chlorophenyl)methyl]-6-oxo-2-phenyl-1H-pyridine-3-carboxylate |
NA |
312400 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
5-benzyl-2-methyl-6-oxo-1H-pyridine-3-carbonitrile |
NA |
128300 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
ethyl 2-methyl-5-[(4-methylphenyl)methyl]-6-oxo-1H-pyridine-3-carboxylate |
NA |
172500 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
methyl 5-benzyl-2-methyl-6-oxo-1H-pyridine-3-carboxylate |
NA |
163500 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
5-[(2-chlorophenyl)methyl]-2-methyl-6-oxo-1H-pyridine-3-carbonitrile |
NA |
423200 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
5-[(2,4-dichlorophenyl)methyl]-2-methyl-6-oxo-1H-pyridine-3-carbonitrile |
NA |
280700 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
ethyl 5-[(2,4-dichlorophenyl)methyl]-2-methyl-6-oxo-1H-pyridine-3-carboxylate |
NA |
172130 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE3A |
8-Fluoro-6-methoxy-3-methyl-1-(2-methylpyridin-3-yl)pyrazolo[3,4-c]cinnoline |
NA |
111900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
3-Methoxy-2-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)phenoxy]methyl]quinoline |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE3A |
4-[5-(4-Chloro-phenyl)-3-methyl-3H-[1,3,4]thiadiazol-(2Z)-ylideneamino]-phenol |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |