| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE3A |
3-(4-Imidazol-1-ylphenyl)-4-methyl-1,4-dihydropyrazol-5-one |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4-Ethyl-3-(4-imidazol-1-ylphenyl)-1,4-dihydropyrazol-5-one |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4,4-diethyl-3-(4-imidazol-1-ylphenyl)-1H-pyrazol-5-one |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4,4-dimethyl-3-(4-pyridin-4-ylphenyl)-1H-pyrazol-5-one |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2,4-dihydro-5-[4-(1H-imidazol-1-yl)phenyl]-3H-pyrazol-3-one |
NA |
590000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
4-cyclopentyl-6,7-dimethoxy-1-methyl-2H-isoquinolin-3-one |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2-(4-Imidazol-1-ylanilino)-1,4-dihydroimidazol-5-one |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
6-(1,4,5,6-Tetrahydro-6-oxopyridazin-3-yl)-2H-benzo[b][1,4]oxazin-3(4H)-one |
NA |
630000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
1H-Imidazo(4,5-b)pyridine, 2-(2,4-dimethoxyphenyl)- |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
1H-Purine-2,6-dione, 3,7-dihydro-7-(2-hydroxypropyl)-1,3-dimethyl-, (S)- |
1200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
1H-Purine-2,6-dione, 3,7-dihydro-7-(2-hydroxypropyl)-1,3-dimethyl-, (R)- |
1100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
2-[(1-hydroxy-3H-2,1-benzoxaborol-5-yl)oxy]-6-(trifluoromethyl)quinoline |
NA |
8130000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
Ici 58301 |
217000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
Theophylline |
NA |
240000|360000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE3A |
3-(6-Chloropyridazin-3-yl)-2-isopropylpyrazolo[1,5-a]pyridine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PDE3A |
4-Methylquinazolin-2(1H)-one |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE3A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| PDE3A |
Ibudilast |
NA |
299000 |
NA |
NA |
NA |
NA |
BindingDB|GtoPDB|PubChem|TTD |
| PDE3A |
Amrinone |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE3A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |