Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| PDE1B | 6-(3-Imidazol-1-yl-phenyl)-4,5-dihydro-2H-pyridazin-3-one | NA | 930000 | NA | NA | NA | NA | BindingDB |
| PDE1B | 6-(4-(1H-Imidazol-1-yl)phenyl)-5-methylpyridazin-3(2H)-one | NA | 660000 | NA | NA | NA | NA | BindingDB |
| PDE1B | 1H-Imidazo(4,5-b)pyridine, 2-(2,4-dimethoxyphenyl)- | NA | 265000 | NA | NA | NA | NA | BindingDB |
| PDE1B | Ici 58301 | 717000 | NA | NA | NA | NA | NA | BindingDB |
| PDE1B | Theophylline | NA | 320000|356000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE1B | Cilostazol | NA | 1000000 | NA | NA | NA | NA | PubChem |
| PDE1B | 4,5-dihydro-6-(4-(imidazol-1-yl)phenyl)-5-methyl-3(2H)-pyridazinone | NA | 3400000 | NA | NA | NA | NA | BindingDB |
| PDE1B | Amrinone | NA | 1000000|300000 | NA | NA | NA | NA | PubChem |
| PDE1B | Milrinone | NA | 198000|310000|340000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE1B | 4-(4-Imidazol-1-yl-phenyl)-4a,5,6,7,8,8a-hexahydro-2H-phthalazin-1-one | NA | 380000|550000 | NA | NA | NA | NA | BindingDB |
| PDE1B | 5-(4-Imidazol-1-yl-phenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydro-pyridine-3-carbonitrile | NA | 130000 | NA | NA | NA | NA | BindingDB |
| PDE1B | 1-butyl-3-propyl-5,7-dihydro-4H-purine-2,6-dione | NA | 149000 | NA | NA | NA | NA | BindingDB |
| PDE1B | Crisaborole | NA | 17900000 | NA | NA | NA | NA | BindingDB|PubChem |
| PDE1B | Roflumilast | NA | 200000 | NA | NA | NA | NA | PubChem |
| PDE1B | 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone | NA | 250000 | NA | NA | NA | NA | BindingDB |
| PDE1B | Rolipram | NA|200000 | 200000|NA | NA | NA | NA | NA | PubChem |
| PDE1B | Enoximone | NA | 1000000 | NA | NA | NA | NA | PubChem |
| PDE1B | Imazodan | NA | 3400000 | NA | NA | NA | NA | BindingDB |
| PDE1B | Filaminast | NA | 190000 | NA | NA | NA | NA | BindingDB |
| PDE1C | Theophylline | NA | 320000|356000 | NA | NA | NA | NA | PubChem |