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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PAOX 3-N-[[2-(3,5-dimethylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(4-fluorophenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(4-tert-butylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(4-Phenylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(4-methylsulfanylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-[4-bromo-2-(trifluoromethyl)phenoxy]phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(3,5-dimethoxyphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX 3-N-[[2-(2,3-dimethylphenoxy)phenyl]methyl]-1H-1,2,4-triazole-3,5-diamine NA 200000 NA NA NA NA TTD
PAOX N-(10-Amino-decyl)-acetamide 110000 NA NA NA NA NA TTD
PAOX N*1*-Prop-2-ynyl-butane-1,4-diamine 425000 NA NA NA NA NA TTD
PAOX N-Methyl-N''-prop-2-ynyl-butane-1,4-diamine 310000 NA NA NA NA NA TTD
PAOX N1-Acetylspermidine 1370000 NA NA NA NA NA PubChem|TTD
PARG 3-(cyclohexylmethyl)-1-methyl-N-(1-methylcyclopropyl)-2,4-dioxoquinazoline-6-sulfonamide NA NA NA 150000 NA NA TTD
PARG N-tert-butyl-1,3-dimethyl-2,4-dioxoquinazoline-6-sulfonamide NA NA NA 110000 NA NA TTD
PARG 3-[(9,10-Dioxoanthracen-2-yl)sulfonylamino]propanamide NA NA NA 150000 NA NA TTD
PARG 2-[(9,10-Dioxoanthracen-2-yl)sulfonylamino]acetamide NA NA NA 150000 NA NA TTD
PARG N-(1-methylcyclopropyl)naphthalene-2-sulfonamide NA NA NA 150000 NA NA TTD
PARG N-(1-methoxy-2-methylpropan-2-yl)-9,10-dioxoanthracene-2-sulfonamide NA NA NA 150000 NA NA TTD
PARG N-ethyl-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-sulfonamide NA NA NA 150000 NA NA TTD
PARG N-ethyl-9,10-dioxo-9,10-dihydroanthracene-2-sulfonamide NA NA NA 110000 NA NA TTD