| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PADI4 |
Doxycycline |
NA|630000 |
860000|NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
Tetracycline |
NA |
780000 |
NA |
NA |
NA |
NA |
PubChem |
| PADI4 |
Chlortetracycline |
540000|110000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PADI4 |
Minocycline |
NA|540000|180000 |
620000|NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PADI4 |
(2S)-5-[(1-amino-2-fluoroethylidene)amino]-2-(benzenesulfonamido)pentanamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
N-[(2S)-1-amino-5-[(1-amino-2-fluoroethylidene)amino]-1-oxopentan-2-yl]-1H-imidazole-5-carboxamide |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
2-fluoro-N-propylacetamidine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
N'-benzyl-2-fluoroethanimidamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
2-fluoro-N'-phenylethanimidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
N-[(2S)-1-amino-3-[3-[(1-amino-2-fluoroethylidene)amino]phenyl]-1-oxopropan-2-yl]benzamide |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
N-[(1S)-2-amino-1-[3-[(1-amino-2-fluoroethylidene)amino]phenyl]-2-oxoethyl]benzamide |
NA |
2100000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
N-[(2S)-1-amino-3-[4-[(1-amino-2-fluoroethylidene)amino]phenyl]-1-oxopropan-2-yl]benzamide |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
N-[(2S)-1-amino-3-[4-[[(1-amino-2-fluoroethylidene)amino]methyl]phenyl]-1-oxopropan-2-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
N-[4-[(1-amino-2-fluoroethylidene)amino]butyl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
N'-[4-(benzenesulfonamido)butyl]-2-fluoroethanimidamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PADI4 |
Trimethoprim |
NA |
7500000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PADI4 |
(4S,4aS,5aS,6S,12aS)-7-chloro-4-(dimethylamino)-6,10,12a-trihydroxy-6-methyl-1,3,11,12-tetraoxo-4a,5,5a,11a-tetrahydro-4H-tetracene-2-carboxamide |
110000|540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
5,5-Dimethyl-3-(piperazin-1-ylmethyl)imidazolidine-2,4-dione |
183000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PADI4 |
1,1'-((1S,2S,3R,4S,5S,6R)-4-(((2R,3R,4R,5S)-3-(((2S,3S,4S,5R,6S)-4,5-Dihydroxy-6-(hydroxymethyl)-3-(methylamino)tetrahydro-2H-pyran-2-yl)oxy)-4-formyl-4-hydroxy-5-methyltetrahydrofuran-2-yl)oxy)-2,5,6-trihydroxycyclohexane-1,3-diyl)diguanidine |
NA|560000 |
1800000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| PADI4 |
(2S,4R)-N-[(1S,2S)-2-chloro-1-[(2R,3R,4S,5R,6R)-3,4,5-trihydroxy-2-methyl-6-methylsulfanyloxan-2-yl]propyl]-1-methyl-4-propylpyrrolidine-2-carboxamide |
NA |
5100000 |
NA |
NA |
NA |
NA |
BindingDB |